Introduction
The regulation of actomyosin contractility plays a key role in
various cellular functions, such as smooth-muscle contraction
(Tan et al., 1992; Fukata et al., 2001), stress fiber and focal
adhesion formation (Tan et al., 1992; Chrzanowska-Wodnicka
and Burridge, 1996), neuronal morphogenesis (Lin et al.,
1996; Amano et al., 1998; Wylie et al., 1998), cytokinesis (De
Lozanne and Spudich, 1987; Komatsu et al., 2000) and
apoptotic membrane blebbing (Mills et al., 1998). In both
smooth muscle and nonmuscle cells, actomyosin contractility
is primarily regulated by phosphorylation of the regulatory
light chain of myosin II (MLC) (Tan et al., 1992).
Phosphorylation of MLC at Thr18 and Ser19 enhances the
actin-activated myosin motor activity (Kamm and Stull,
1989), whereas phosphorylation at Ser1/2 and Thr9 by protein
kinase C (PKC) decreases its affinity for actin (Bengur et al.,
1987). Phosphorylation of MLC at Thr18 and Ser19 is
regulated by the MLC kinases and phosphatases. Myosin-
light-chain kinase (MLCK) is responsible for calcium-
dependent MLC phosphorylation at the stimulatory sites
(Kamm and Stull, 1989). Rho kinase (ROCK) can both
inactivate MLC phosphatase by phosphorylating its myosin-
binding subunit (Kimura et al., 1996; Feng et al., 1999;
Kawano et al., 1999) and directly phosphorylate MLC at
MLCK site (Amano et al., 1996; Ueda et al., 2002). The p21-
activated kinase was also reported to increase MLC
phosphorylation in certain cell types (Kiosses et al., 1999;
Sells et al., 1999). Through alterations of the MLC
phosphorylation, these kinases and phosphatases regulate
actomyosin contractile forces, profoundly influencing cell
motility and morphology (Wilson et al., 1991; Klemke et al.,
1997; Dong et al., 1998; Fukata et al., 1999).
Contractility of nonmuscle cells is intimately associated
with adhesion and adhesion-dependent signaling. Focal
adhesions are sites of contact between the cell surface and
the extracellular matrix, where the associated stress fibers
terminate. They consist of both structural proteins that link
integrins to the actin cytoskeleton and signaling proteins that
transduce a range of adhesion-dependent signals (Sastry and
Burridge, 2000; Zamir and Geiger, 2001). The assembly and
stabilization of focal adhesions is greatly influenced by
myosin-II-driven contractility. Chemicals that inhibit either
MLC phosphorylation or actin-dependent myosin ATPase
activity cause a rapid loss of both stress fibers and focal
adhesions (Volberg et al., 1994; Chrzanowska-Wodnicka and
Burridge, 1996). Similar effects are observed by dominant-
negative inhibition of myosin IIA heavy chain (Wei and
Adelstein, 2000) or overexpression of caldesmon (Helfman
et al., 1999), a protein that restrains the interactions of
myosin heads with actin filaments. Conversely, activation of
the Rho/ROCK pathway stimulates the formation of both
stress fibers and their associated focal adhesions in a
contractility-dependent manner (Amano et al., 1997; Uehata
et al., 1997).
MLC phosphorylation is also involved in apoptosis.
Death-associated protein kinase (DAP kinase) is a
4777
Death-associated protein kinase (DAP kinase) is a pro-
apoptotic, calcium/calmodulin-dependent serine/threonine
kinase. Here, we report that DAP kinase phosphorylates
the regulatory light chain of myosin II (MLC) both in vitro
and in vivo, and that this phosphorylation occurs
preferentially at residue Ser19. In quiescent fibroblasts,
DAP kinase stabilizes stress fibers through phosphorylation
of MLC, but it is dispensable for the formation of
peripheral microfilament bundles. This cytoskeletal effect
of DAP kinase occurs before the onset of apoptosis and does
not require an intact death domain. In addition, DAP
kinase is required for serum-induced stress-fiber
formation, which is associated with the upregulation of its
catalytic activity. Despite being both sufficient and
necessary for the assembly or maintenance of stress fibers,
DAP kinase is incapable of stimulating the formation of
focal adhesions in quiescent cells. Moreover, it promotes the
disassembly of focal adhesions but not stress fibers in cells
receiving serum factors. Together, our results identify a
novel and unique function of DAP kinase in the uncoupling
of stress fibers and focal adhesions. Such uncoupling would
lead to a perturbation of the balance between contractile
and adhesion forces and subsequent cell detachment, which
might contribute to its pro-apoptotic activity.
Key words: DAP kinase, Myosin phosphorylation, Stress fibers,
Focal adhesions, Apoptosis
Summary
Uncoordinated regulation of stress fibers and focal
adhesions by DAP kinase
Jean-Cheng Kuo
1
, Jia-Ren Lin
1
, James M. Staddon
2
, Hiroshi Hosoya
3
and Ruey-Hwa Chen
1,
*
1
Institute of Molecular Medicine, College of Medicine, National Taiwan University, Taipei, Taiwan
2
Eisai London Research Laboratories, University College London, London, UK
3
Department of Biological Science, Graduate School of Science, Hiroshima University, Higashi-Hiroshima, Hiroshima, Japan
*Author for correspondence (e-mail: rhchen@ha.mc.ntu.edu.tw)
Accepted 22 July 2003
Journal of Cell Science 116, 4777-4790 © 2003 The Company of Biologists Ltd
doi:10.1242/jcs.00794
Research Article