335 © Springer Nature Singapore Pte Ltd. 2019
A. Misra, A. Shahiwala (eds.), Novel Drug Delivery Technologies,
https://doi.org/10.1007/978-981-13-3642-3_10
A. Desai · M. Shukla · F. Maulvi · K. Ranch (*)
Department of Pharmaceutics, Maliba Pharmacy College, Uka Tarsadia University,
Surat, Gujarat, India
10
Ophthalmic and Otic Drug
Administration: Novel Approaches
and Challenges
Ankita Desai, Manish Shukla, Furqan Maulvi,
and Ketan Ranch
Contents
10.1 Ocular Drug Delivery 337
10.1.1 General Introduction to Ocular Drug Delivery 337
10.1.1.1 Mechanism of Ocular Drug Absorption 337
10.1.1.2 Routes of Ocular Drug Delivery-Conventional vs. Novel Routes 338
10.1.1.3 Challenges for Ophthalmic Drug Delivery Systems 339
10.1.2 Important Factors for Ophthalmic Drug Delivery Systems 340
10.1.2.1 Barriers to Restrict Intraocular Drug Transport/Factors Affecting
Intraocular Bioavailability 340
10.1.2.2 Physicochemical Property of Drug Candidate 341
10.1.2.3 Formulation Factors 342
10.1.3 Ideal Characteristics of Ocular Drug Delivery Systems 344
10.1.4 Conventional Dosage Forms for Ocular Drug Delivery with Their
Limitations 344
10.1.4.1 Topical Eye Drops 345
10.1.4.2 Emulsions 346
10.1.4.3 Suspensions 346
10.1.4.4 Semisolid Ophthalmic Drug Forms: Eye Ointments 347
10.1.5 Novel Strategies/Approaches to Enhance Ocular Bioavailability 347
10.1.5.1 Nanotechnology-Based Ocular Drug Delivery 347
10.1.5.2 Polymer Gels 352
10.1.5.3 Other Drug Delivery Systems 355
10.1.6 New Trends/Emerging Technologies for Ocular Drug Delivery 357
10.1.6.1 Punctal Plug Delivery System (PPDS) or Evolute® 357
10.1.6.2 DelSiTech® 358
10.1.6.3 OpsiSporin 360
10.1.6.4 ForSight VISION5® 361
10.1.6.5 OcuSurf™ 362
10.1.7 Biodegradable Polymers for Ophthalmic Applications 364
10.1.7.1 Natural Biodegradable Polymers 364