Vol 11, Issue 12, 2018
Online - 2455-3891
Print - 0974-2441
FUSOGENIC LIPOSOME FOR THE TREATMENT OF FUNGAL
MENINGITIS: AN OVERVIEW
IRENE SUSAN ALEX, JENEETTA JOSE, RAHUL R, ANJU GOPAL, ANU PRIYA*
Department of Pharmaceutics, Amrita School of Pharmacy, Amrita Institute of Medical Sciences and Research Centre, Amrita Vishwa
Vidyapeetham, Kochi, Kerala, India. Email: anupriya@aims.amrita.edu
Received: 23 April 2018, Revised and Accepted: 11 August 2018
ABSTRACT
Fungal meningitis is an infection which is caused by fungus which spreads through the blood to the spinal cord. People with weakened immunity
get this disease easily like persons with AIDs, etc. To make sure the disease is fungal meningitis, a sample is taken from the cerebrospinal fluid
and it is sent to the laboratory. Usually, fungal meningitis is not mediated from person to person, but it is caused when a fungi are inhaled from
the surrounding and spread into the blood to the central nervous system. Normally medications such as vaccines, IV, and oral suspensions are
given to the people for curing fungal meningitis. Commonly used drugs are Amphotericin B and fluconazole oral suspension. Amphotericin B is
an antifungal, antiprotozoal, and hydrophobic drug. However, these drugs cannot give a directly as medication therapy for the patients, because
it offers toxic effect and side effects, absorption rate is slower, and crossing the blood–brain barrier (BBB) is getting difficult. Adverse effects can
be minimized with the application of nanotechnology. Therefore, in human medical services, the availability of molecular nanotechnology will
provide rapid progress. Nanoparticle (NP) systems help to improve the solubility of poorly water-soluble drugs which has been explained using
Noyes–Whitney equations. Nanoparticles offers several advantages as a drug delivery system, such as better drug bioavailability, reduction of
dosing frequency enables them for the betterment of diseases, can cross the BBB, and it is very cost-effective. Types of NP include polymeric NP,
carbon nanotubes, metallic structures, nanocrystals, and fusogenic liposomes. Fusogenic liposomes are a peculiar class of phospholipid vesicles. The
fusogenic liposomes can deliver encapsulated NP into the targeted sites and also can cross the BBB. On comparing with cationic liposomes, fusogenic
liposomes are more effective as well as rapid in the drug delivery.
Keywords: Fungal meningitis, Nanotechnology, Liposomes, Fusogenic liposomes.
INTRODUCTION
Among different types of fungal infections, one of the types is fungal
meningitis. Fungal meningitis is caused due to the inhalation of fungus
spores or localized colonization of the skin. Cryptococcus fungus is
the main causative organism of fungal meningitis; it is also caused
by other organisms. The organisms are generally breathed in and
afterward spread into the blood and to the focal sensory system yet it
is not spread starting with one individual then onto the next [1]. The
growths can likewise be specifically embedded into the focal sensory
system by medicinal methods or can be entered from a tainted site
close to the focal sensory system which can cause meningitis. Any
treatment that may debilitate the insusceptible framework may
prompt high hazard components of contagious meningitis. The other
hazard factors incorporate surgical methods that are managed with
no sterility and will acquaint the growths with the focal anxious.
Cerebral pain, solid neck, queasiness, heaving, photophobia, and
adjusted mental status are its primary side effects. This is diagnosed
by blood and culture of cerebrospinal fluid. The most effective thing
to protect children from meningitis is to provide vaccines that protect
against most forms of meningitis and septicaemia [2]. Commonly
IV antifungal drugs and oral suspensions such as fluconazole and
Amphotericin B drugs are given for this treatment. Different drug
delivery systems have been developed with the help of nanoparticles
(NPs) [3].
PATHOGENESIS
The key step for a pathogen to infect the brain and cause
meningitis is to cross the blood–brain barrier (BBB), an interface
that separates the peripheral circulation and central nervous
system [4].
BASIC PATHOLOGY OF FUNGAL MENINGITIS [5]
© 2018 The Authors. Published by Innovare Academic Sciences Pvt Ltd. This is an open access article under the CC BY license (http://creativecommons.
org/licenses/by/4. 0/) DOI: http://dx.doi.org/10.22159/ajpcr.2018.v11i12.26852
Review Article