healthcare
Article
The Role of CDK4 in the Pathogenesis of Pancreatic Cancer
Emily Jiggens
1
, Maria Mortoglou
1
, Guy H. Grant
2
and Pinar Uysal-Onganer
1,
*
Citation: Jiggens, E.; Mortoglou, M.;
Grant, G.H.; Uysal-Onganer, P. The
Role of CDK4 in the Pathogenesis of
Pancreatic Cancer. Healthcare 2021, 9,
1478. https://doi.org/10.3390/
healthcare9111478
Academic Editors: Nur Mohammad
Hassan, Rahena Akhter and
Paolo Cotogni
Received: 20 August 2021
Accepted: 28 October 2021
Published: 30 October 2021
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4.0/).
1
Cancer Research Group, School of Life Sciences, University of Westminster, London W1W 6UW, UK;
w1712684@my.westminster.ac.uk (E.J.); w1754188@my.westminster.ac.uk (M.M.)
2
Department of Life Sciences, University of Bedfordshire, Park Square, Luton LU1 3JU, UK;
guy.grant@beds.ac.uk
* Correspondence: p.onganer@westminster.ac.uk; Tel.: +44-(0)207-911-5151 (ext. 64581)
Abstract: Pancreatic cancer (PC) continues to have the lowest overall survival and the lack of
effective early diagnosis. Cyclin-dependent kinase 4 (CDK4) plays a fundamental role in the orderly
progression of the cell cycle, binding to cyclin D to promote the progression through the G1/2
transition. The inhibition of CDK4/6 has therefore gained substantial interest in the hope of new
and effective therapeutics in multiple cancers, such as advanced metastatic breast cancer. While
the use of these agents is encouraging, their potential is yet to be fully explored. In this study we
used the GLOBOCAN database to understand the most recent epidemiology of PC, Human Protein
Atlas and KEGG to highlight the role, prevalence, and significance on patient survival of CDK4 in
PC. We found that CDK4 cannot be used as prognostic in PC and no significant differences were
observed between CDK4 expression and the patient’s clinical status, though larger studies, especially
concerning CDK4 protein expressions, are required for a more thorough understanding. The use
of CDK4/6 inhibitors in PC is still in clinical trials. However, due to only modest improvements
observed in the use of single-agent therapies, efforts have focused on combinatorial approaches.
Keywords: pancreatic cancer; CDK4; CDK4/6 inhibitor; epidemiology
1. Introduction
Pancreatic Cancer (PC) is a highly aggressive malignancy, which continues to have the
lowest overall 1- and 5-year patient survival rates amongst all cancer sites in the United
Kingdom, at 25% and 7%, respectively [1]. While surgical resection remains the only
curative treatment available, 80–85% of tumours are diagnosed at late and unresectable
stages, with evidence of locally advanced or metastatic disease. For the small proportion
of patients that do qualify for surgical care, survival rates are modest - despite numerous
benefits observed when studying the early detection of PC [2] - and patients frequently
suffer from local recurrence, metachronous metastasis and high tumour chemoresistance
following resection, seen in up to 80% of cases [3]. Despite advances in diagnostic tech-
nology, the high frequency of late-stage diagnoses, and the associated poor prognosis,
is largely attributable to the non-specific early-stage symptoms, the lack of specific and
sensitive biomarkers, and the retroperitoneal position of the pancreas that restricts the
accessibility of routine checks [4].
Pancreatic ductal adenocarcinoma (PDAC) is an invasive pancreatic epithelial neo-
plasm with glandular differentiation and is the most prevalent histological subtype of
PC, accounting for approximately 85% of pancreatic tumours; the terms PC and PDAC
are often used synonymously. In recent studies, several subtypes of PDAC have been
defined following gene expression analysis. The implications they hold for future precision
medicine and targeted patient clinical care is promising: results show that the presence of
stromal infiltration improves survival in patients with desmoplastic or stroma-activated
subtypes, whereas basal-like tumours have an unfavourable prognosis and a poor median
overall survival (OS) rate of 10.3 months. However, these lack consensus and a universally
agreed classification system is required for implementation into routine clinical practice [5].
Healthcare 2021, 9, 1478. https://doi.org/10.3390/healthcare9111478 https://www.mdpi.com/journal/healthcare