Epidemiologic Reviews
Copyright © 2001 by the Johns Hopkins University Bloomberg School of Public Health
All rights reserved
Vol. 23, No. 1
Printed in U.S.A.
Potential Agents for Prostate Cancer Chemoprevention
Otis W. Brawley
1
and Shakia T. Barnes
2
INTRODUCTION
Studies of the incidence and mortality of prostate cancer
in various countries suggest that changeable environmental
elements are important in its etiology (1). Several studies
have demonstrated that migration from areas of low risk to
areas of high risk is associated with an increased risk of
prostate cancer in the migrants compared with men remain-
ing in the low-risk country of origin (1). In migration stud-
ies done before the prostate-specific antigen screening era,
Japanese migrants to the United States were shown to have
a marked increase in prostate cancer, although the rates of
Japanese-Americans remain less than those of whites (2).
Prostate cancer incidence rates are very low in eastern
Europe and Russia, but Polish migrants to the United States
acquire higher rates upon migration.
While population studies do suggest that there may be a
genetic component to some prostate cancers, there are
likely to be numerous environmental components to
prostate carcinogenesis and prostate cancer prevention (3).
Nutritional factors in defined populations, especially in
those with high animal fat and high dairy intake, have been
correlated with a greater risk of disease (4). It has been
suggested that populations with higher circulating levels of
androgens and insulin-like growth factors tend to have
higher risk of prostate cancer (5, 6). Both circulating
androgens and insulin-like growth factor levels are associ-
ated with diet (7, 8). In at least one case-control study with
age-adjusted analyses, there were positive associations of
prostate cancer (all stages combined) risk with total energy
intake as well as intake of total fat (saturated and monoun-
saturated) (9). There are also correlations between popula-
tions with higher consumption of selenium and vitamin E,
fructose/fruits, and tomatoes and lower risk of prostate
cancer (10). These observations combined with an
improved understanding of the biology of prostate cancer
Received for publication December 5, 2000, and accepted for
publication May 25, 2001.
Abbreviations: NSAIDs, non-steroidal anti-inflammatory drugs;
SELECT, Selenium and Vitamin E Comparison Trial.
1
Winship Cancer Institute, Emory University School of Medicine,
Atlanta, GA.
2
Office of the Director, National Cancer Institute, Bethesda, MD.
Reprint requests to Dr. Otis W. Brawley, Winship Cancer Institute,
Emory University School of Medicine, Emory Clinic Building B, Suite
B4100,1365-B Clifton Road, Atlanta, GA 30322 (e-mail: otis_brawley@
emory.org).
provide numerous leads in the effort to find workable
prostate cancer chemoprevention (11).
CONCEPT OF CHEMOPREVENTION
Chemoprevention is the administration of agents to pre-
vent induction and inhibit or delay progression of cancers.
Important to chemoprevention is the fact that carcinogene-
sis is a process over time involving cellular growth and
division. Inhibition of or slowing this process can poten-
tially prevent cancers from becoming clinically significant
(12). While chemoprevention of cancer is a relatively new
concept, the chemoprevention of other diseases is common
although often not called chemoprevention. The prevention
of heart disease with lipid lowering drugs is widely
accepted, as is the prevention of tooth decay with flouride
or prevention of osteoporosis in postmenopausal women
with estrogen (13). These are all examples of chemopre-
vention of disease.
Chemoprevention involves the treatment of healthy
subjects. As such, chemopreventive agents must have low
toxicity in order to be clinically useful (14-16). Because
their purpose is to keep something from occurring, defin-
itive clinical studies to demonstrate their efficacy are
necessarily randomized, blinded, long-term, and large in
size.
It has been suggested that androgen is an important pro-
moter of prostate cancer. It has long been appreciated that
prostate cancer is an androgen-driven illness. Removal of
androgenic stimulation has been used to treat metastatic
disease for some time (17). Populations with impaired
androgen metabolism, such as congenital 5oc-reductase defi-
ciency, do not develop prostate cancer. There is also the sug-
gestion that populations with higher circulating levels of
androgen or higher sensitivity to androgens are at greater
risk of prostate cancer (18, 19).
Oxidative stress has been proposed as a promoter of the
process of carcinogenesis. Oxidation can lead to genetic
mutations which can, in turn, lead to malignancy.
Antioxidants have been suggested as potential preventative
agents for a number of cancers (4).
DIET AND PROSTATE CANCER
Dietary intervention is not classically considered
chemoprevention, but it could be very important in the
prevention of prostate cancer. Some dietary elements may
cause prostate cancer, whereas elements in other diets may
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