Pawar et al Journal of Drug Delivery & Therapeutics. 2019; 9(6-s):216-228
ISSN: 2250-1177 [216] CODEN (USA): JDDTAO
Available online on 15.12.2019 at http://jddtonline.info
Journal of Drug Delivery and Therapeutics
Open Access to Pharmaceutical and Medical Research
© 2011-18, publisher and licensee JDDT, This is an Open Access article which permits
unrestricted non-commercial use, provided the original work is properly cited
Open Access Review Article
Importance of Nanocarriers and Probiotics in the Treatment of Ulcerative
Colitis
Amandeep Singh
1 2
*, Kirandeep Kaur
1
, Veerpal Kaur
1
, Gurmeet Singh
1
, Uttam Kumar Mandal
2
, Neeraj
Mishra
3
, Raj Kumar Narnag
1
1
Department of Pharmaceutics, ISF College of Pharmacy, Moga-142001, Punjab, India
2
Department of Pharmaceutical Sciences and Technology, Maharaja Ranjit Singh Punjab Technical University, Bathinda- 151001, Punjab, India.
3
Department of Pharmaceutics, Amity Institute of Pharmacy, Gwalior, Madhya Pradesh, India
ABSTRACT
Ulcerative colitis (UC) is an inflammatory chronic disease primarily affecting the colonic mucosa; the extent and severity of colon involvement
are variable. In its most limited form, it may be restricted to the distal rectum, while in its most extended form the entire colon is involved.
Ulcerative colitis is identified by mucus diarrhea, tenesmus, bowel distension, and anemia. 5-aminosalicylic acid drugs, steroids, and
immunosuppressant are used for therapy of ulcerative colitis. The annual occurrence of disease in Asia, America, and Europe was estimated to
be 6.3, 19.2 and 24.3 per 100,000 people-years. The main challenges in the management of the diseaseare drug-related side-effects and local
targeting. To overcome these challenges probiotics and micro and Nano particulate system auspicious approaches to overcome drug-related
adverse side effect and local targeting. Upon ingestion, the probiotics can result in health beneficial effects. Probiotics are mainly used as gut
modulators but are also now days explored for their use in ulcerative colitis. Micro and Nano particulate drug delivery system have been
achieving huge importance for targeting of the drug to colon locally at a controlled and sustained rate. The main objective of this article is to
explore probiotics and micro and nano particulate approaches for the suitable targeting and overcome the drug-associated side effect.
Keywords: Inflammatory chronic disease, probiotics, micro and Nano particulate.
Article Info: Received 03 Oct 2019; Review Completed 11 Nov 2019; Accepted 18 Nov 2019; Available online 15 Dec 2019
Cite this article as:
Singh A, Kaur K, Kaur V, Singh G, Mandal UK, Mishra N, Narnag RK, Importance of Nanocarriers and Probiotics in the
Treatment of Ulcerative Colitis, Journal of Drug Delivery and Therapeutics. 2019; 9(6-s):216-228
http://dx.doi.org/10.22270/jddt.v9i6-s.3727
*Address for Correspondence:
Amandeep Singh, Assistant Professor, Department of Pharmaceutics, ISF College of Pharmacy, Moga, Punjab, India Postal Code: 142001.
INTRODUCTION
IBD is a disease of the gastrointestinal tract and it
isidentified by unrestricted inflammation caused by
unsuitable and constant activation of the mucosal immune
system. Ulcerative colitis and Crohn’s disease are the
different types of the inflammatory bowel disease (IBD)
which are very common, with associated significant
morbidity and mortality[1],[2]. While the main reasons are
mostly undetermined of the pathogenesis of IBD but the
factors related to the environment and genetic vulnerability
are found to be associated with it[3].Ulcerative colitis is
chronic inflammatory disorders found in the intestinal tract
that causes life-threatening issue and have an increasing
occurrence worldwide [4]. Small intestine and large intestine
or colon are the major areas involved in the IBD, which are
manifested by the persistent inflammation in certain areas of
mucosa[5]. It is determined by intermittent rectal bleeding,
diarrhoea, rectal urgency and tenesmus[6]. In Western
Europe, Asia and North America, this disease has an annual
occurrence of approximately 24.3 per 100,000 populations
every year, 6.3 per 100,000 per year and 19.2 per 100,000
populations every year, respectively. IBD is becoming a
world disorder because of increasing occurrence and
prevalences of it with respect to time. There is a very lower
occurrence in Africa, South America and Asia[7]. It has been
predicted that more than 1 million individuals suffered from
IBD in the US, out of which, 100,000 are children. IBD is in
5th rank amid the most common gastrointestinal disorder.
Epidemiology
The occurrence and prevalence of ulcerative colitis have
been expanding over time worldwide. Ulcerative colitis is
mainly related to recurrent attacks with complete remission
of symptoms. The increased incidence of the disease is more
(three to six-fold more) in Jewish and it is more common in
Caucasians than in black. In Western Europe occurrence of