polymers
Article
Synthesis and Characterization of a Bioconjugate Based on
Oleic Acid and L-Cysteine
Marco Vizcarra-Pacheco
1
, María Ley-Flores
2
, Ana Mizrahim Matrecitos-Burruel
3
, Ricardo López-Esparza
1
,
Daniel Fernández-Quiroz
4
, Armando Lucero-Acuña
1,4
and Paul Zavala-Rivera
1,4,
*
Citation: Vizcarra-Pacheco, M.;
Ley-Flores, M.; Matrecitos-Burruel,
A.M.; López-Esparza, R.; Fernández-
Quiroz, D.; Lucero-Acuña, A.;
Zavala-Rivera, P. Synthesis and
Characterization of a Bioconjugate
Based on Oleic Acid and L-Cysteine.
Polymers 2021, 13, 1791. https://
doi.org/10.3390/polym13111791
Academic Editors: TriDung Ngo and
Aman Ullah
Received: 13 March 2021
Accepted: 25 May 2021
Published: 29 May 2021
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1
Departamento de Física, Universidad de Sonora, Blvd. Luis Encinas y Rosales S/N, Colonia Centro,
83000 Hermosillo, Sonora, Mexico; marco.vizcarra@unison.mx (M.V.-P.); ricardo.lopez@unison.mx (R.L.-E.);
armando.lucero@unison.mx (A.L.-A.)
2
Pritzker School of Molecular Engineering, The University of Chicago, Chicago, IL 60637, USA;
mleyf@uchicago.edu
3
Departamento de Investigación en Polímeros y Materiales, Universidad de Sonora, Av. Colosio S/N,
Colonia Centro, 83000 Hermosillo, Sonora, Mexico; a213220985@unison.mx
4
Departamento de Ingeniería Química y Metalurgia, Universidad de Sonora, Av. Colosio S/N, Colonia Centro,
83000 Hermosillo, Sonora, Mexico; daniel.fernandez@unison.mx
* Correspondence: paul.zavala@unison.mx
Abstract: One of the main challenges facing materials science today is the synthesis of new biodegrad-
able and biocompatible materials capable of improving existing ones. This work focused on the
synthesis of new biomaterials from the bioconjugation of oleic acid with L-cysteine using carbodi-
imide. The resulting reaction leads to amide bonds between the carboxylic acid of oleic acid and
the primary amine of L-cysteine. The formation of the bioconjugate was corroborated by Fourier
transform infrared spectroscopy (FTIR), Raman spectroscopy, and nuclear magnetic resonance (NMR).
In these techniques, the development of new materials with marked differences with the precursors
was confirmed. Furthermore, NMR has elucidated a surfactant structure, with a hydrophilic part and
a hydrophobic section. Ultraviolet-visible spectroscopy (UV-Vis) was used to determine the critical
micellar concentration (CMC) of the bioconjugate. Subsequently, light diffraction (DLS) was used to
analyze the size of the resulting self-assembled structures. Finally, transmission electron microscopy
(TEM) was obtained, where the shape and size of the self-assembled structures were appreciated.
Keywords: surfactant; oleic acid; L-cysteine; bioconjugation; biomolecule
1. Introduction
This work focused on the synthesis of new biomaterials from the bioconjugation of
oleic acid with L-cysteine using carbodiimide. The process of chemically joining two or
more molecules through a covalent bond with the help of a crosslinking agent is called
bioconjugation. These agents have reactive ends for specific functional groups (primary
amines, sulfhydryls, etc.) [1]. The demand for biocompatible and biodegradable mate-
rials for medical applications has increased the research of new compounds that satisfy
those properties. Within these new compounds, some surfactants could meet these char-
acteristics [2,3]. Surfactants have a characteristic molecular structure comprising a group
(generally a long alkyl chain) with little attraction for the solvent (hydrophobic, if the
solvent is water), together with another group (ionic or non-ionic) that shows a strong at-
traction of the solvent (hydrophilic in aqueous systems). The degree of surface activity and
the type of application depends on the hydrophilic/lipophilic balance (HLB) characteristics
of this amphiphilic structure [4]. The surfactant molecules of renewable raw materials that
mimic natural lipoamino acids are one of the preferred options for food, pharmaceutical,
and cosmetic applications [5]. These surfactants can be obtained from molecules that mimic
natural amphiphilic structures. Based on these considerations, and as part of our study
objective, a surfactant was synthesized from oleic acid and cysteine (lipoamino acids). The
Polymers 2021, 13, 1791. https://doi.org/10.3390/polym13111791 https://www.mdpi.com/journal/polymers