Research Article
Antimalarial Properties of Aqueous Crude
Extracts of Gynostemma pentaphyllum and Moringa oleifera
Leaves in Combination with Artesunate in
Plasmodium berghei-Infected Mice
Voravuth Somsak, Preeyanuch Borkaew, Chokdee Klubsri, Kittiyaporn Dondee,
Panatda Bootprom, and Butsarat Saiphet
Department of Clinical Chemistry, Faculty of Medical Technology, Western University, Kanchanaburi 71170, Tailand
Correspondence should be addressed to Voravuth Somsak; voravuthsomsak@gmail.com
Received 9 August 2016; Accepted 20 October 2016
Academic Editor: Sukla Biswas
Copyright © 2016 Voravuth Somsak et al. Tis is an open access article distributed under the Creative Commons Attribution
License, which permits unrestricted use, distribution, and reproduction in any medium, provided the original work is properly
cited.
Due to the emergence and spread of malaria parasite with resistance to antimalarial drugs, discovery and development of new,
safe, and afordable antimalarial are urgently needed. In this respect, medicinal plant extracts are targets to optimize antimalarial
actions and restore efcacy of standard antimalarial drugs. Te present study was aimed at determining the antimalarial activities of
Gynostemma pentaphyllum and Moringa oleifera leaf extracts in combination with artesunate against Plasmodium berghei-infected
mice. P. berghei ANKA maintained by serial passage in ICR mice were used based on intraperitoneal injection of 1 × 10
7
parasitized
erythrocytes and subsequent development of parasitemia. Tese infected mice were used to investigate the antimalarial activity of
artesunate (6 mg/kg) in combination with 500, 1,000, and 2,000 mg/kg of G. pentaphyllum and M. oleifera leaf extracts using 4-day
suppressive test. It was found that these extracts showed signifcant ( < 0.05) antimalarial activity in dose-dependent manner
with percentage of suppression of 45, 50, and 55% for G. pentaphyllum leaf extract and 35, 40, and 50% for M. oleifera leaf extract.
Additionally, artesunate combined with these extracts presented higher antimalarial activity, compared to extract treated alone with
percentage of suppression of 78, 91, and 96% for G. pentaphyllum leaf extract and 73, 82, and 91% for M. oleifera leaf extract. Te
results indicated that combination treatment of G. pentaphyllum or M. oleifera leaf extracts with artesunate was able to increase the
antimalarial activity by using low dose of artesunate. Hence, these results justifed the combination of these extracts and artesunate
in antimalarial herbal remedies.
1. Introduction
Malaria is a major parasitic disease with high mortality
and morbidity, especially in the sub-Saharan Africa, Latin
America, and Asia. About 3 billion people worldwide are
exposed annually, with 1.2 billion at high risk, and some
200 million developed symptomatic malaria. Moreover, it
was estimated that 1 million deaths have occurred in the
world [1]. Tis disease is caused by malarial protozoa parasite
from genus Plasmodium and transmitted by female Anopheles
mosquito. Due to the lack of efective vaccine to prevent
malaria, the global strategy for malaria mainly focuses on case
management through provision of antimalarial drugs which
are capable of reducing or eliminating malaria parasites.
Unfortunately, malaria parasite has developed resistance to
drugs used in malarial therapy except the artemisinin [2].
However, artemisinin produces fast recrudescence when used
alone due to its short half-life. Hence, artemisinin used
in combination with other antimalarials, a combination
known as artemisinin-combination therapy (ACT), has been
recommended [3]. In addition, resistance of mosquitoes to
insecticides has led to an increase in severe malaria, com-
plicating the eradication of the disease, and the resurgence
of malaria [4]. Moreover, many antimalarials in use today
have high toxicity that exposes patients’ health expenditure
[5]. In this respect, medicinal plant extracts are potential
Hindawi Publishing Corporation
Journal of Tropical Medicine
Volume 2016, Article ID 8031392, 6 pages
http://dx.doi.org/10.1155/2016/8031392