Mutation Research, 263 (1991) 115-117
© 1991 ElsevierSciencePublishers B.V. 0165-7992/91/$03.50
ADONIS 016579929100049F
MUTLET 0498
115
Activity of aniline in the mouse bone marrow micronucleus assay
J. Ashby 1, D.A. Vlachos2 and H. TinwelP
11C1 Central Toxicological Laboratory, Alderley Park, Macclesfield, Ches. SKIO 4TJ (Great Britain) and 2 Ciba-Geigy Corporation,
Agricultural Division, Greensboro, N C 27419 (U.S.A.)
(Received28 January 1991)
(Accepted 7 February 1991)
Keywords: Aniline; Mouse; Bone-marrow MN assay
Summary
Aniline gave a positive response in the mouse bone marrow micronucleus assay 24 h after the second of
two intraperitoneal injections of 80% of the median lethal dose (MLD). Negative results were observed at
lower dose levels and at earlier and later sampling times. The significance of this unique activity profile is
discussed within the context of the non-carcinogenicity of aniline to the mouse.
Aniline is carcinogenic to the rat but not the
mouse (Anon., 1978). It is reported also to give a
positive test response in a rat bone-marrow
micronucleus assay (George et al., 1990). The
possible activity of aniline in a mouse bone-
marrow micronucleus assay therefore became of
particular interest. This interest was enhanced by
our recent observation of negative rat and mouse
bone-marrow micronucleus assay data for the po-
tent rat/mouse carcinogen 2-methoxyaniline (o-
anisidine, Ashby et al., 1991). Both chemicals are
biologically available as evidenced by their induc-
tion of methaemoglobinaemia (cyanosis) in both
species of test animal (Anon., 1978; Ashby et al.,
1991).
Correspondence: Dr. J. Ashby, ICI Central Toxicology
Laboratory, Alderley Park, Macclesfield, Ches. SKI0 4TJ
(Great Britain).
Materials and methods
Chemicals. Aniline was re-distilled from
AnalaR grade material (BDH). Cyclophosphamide
(CP) was obtained from the Sigma Chemical Com-
pany, Poole, Dorset. Each was dissolved in sterile
deionized water and administered to mice by in-
traperitoneal injection (10 ml/kg bodyweight),
Micronucleus assays. Bone-marrow smears
were prepared and stained with acridine orange as
described earlier (Tinwell and Ashby, 1989). 2000
polychromatic erythrocytes (PE) were assessed for
micronucleated PE (MPE) on a single slide
prepared from each animal. The ratio of PE to nor-
mocytes (NE) was determined among 1000
erythrocytes on the same slide.
Animals. Male CBA mice aged 8-11 weeks