Sumerianz Journal of Medical and Healthcare, 2021, Vol. 4, No. 2, pp. 109-113
ISSN(e): 2663-421X, ISSN(p): 2706-8404
Website: https://www.sumerianz.com
DOI: https://doi.org/10.47752/sjmh.42.109.113
© Sumerianz Publication
CC BY: Creative Commons Attribution License 4.0
Original Article Open Access
*Corresponding Author
109 109
Manufacture of Hard Gelatin Capsules From a Lyophilisate of the Morus
Nigra Fruit
Sandra Isabel Hernández-González
Laboratorio B de Investigación, Facultad de Ciencias Químicas Campus Gómez Palacio, Universidad Juárez del Estado de
Durango, Mexico
Jesús Iván García-Castañeda
Laboratorio B de Investigación, Facultad de Ciencias Químicas Campus Gómez Palacio, Universidad Juárez del Estado de
Durango, Mexico
José de Jesús Alba-Romero
Laboratorio B de Investigación, Facultad de Ciencias Químicas Campus Gómez Palacio, Universidad Juárez del Estado de
Durango, Mexico
Aurora Martínez-Romero
*
Laboratorio B de Investigación, Facultad de Ciencias Químicas Campus Gómez Palacio, Universidad Juárez del Estado de
Durango, Mexico
Email: aurora.martinez@ujed.mx
Rodolfo Gerardo Chew-Madinaveitia
Instituto Tecnológico de Torreón. Coahuila, Mexico
José Luis Ortega-Sanchez
Unidad Regional Universitaria de Zonas Áridas. Universidad Autónoma Chapingo, Mexico
Article History
Received: April 22, 2021
Revised: May 27, 2021
Accepted: June 4, 2021
Published: June 7, 2021
Abstract
Morus nigra L. (M. nigra L.) belongs to the Moraceae family. Traditional medicine for its physicochemical properties.
To evaluate the physicochemical composition and pharmaceutical stability of hard gelatin capsules of the freeze-dried
fruit of M. nigra L. The content of total phenols (CFT) and antioxidant capacity (CA) were evaluated by
spectrophotometry, the content of ash, moisture, protein, fat and fiber were determined according to their own standard.
The CFT and CA were 25.4 mg gallic acid equivalents/g of sample, and 74.1% inhibition, respectively. On the other
hand, the values of ash, moisture, protein, fat and fiber were 4.2%, 7.9%, 3.9%, 0.5% and 3.6%, respectively.
Lyophilized M. nigra fruit may be a novel candidate for the development of gelatin hard capsules and other new
pharmaceutical products.
Keywords: Physicochemical composition; Pharmaceutical stability; M. nigra L.
1. Introduction
Morus nigra L. (Moraceae family), also known as blackberry, is one of the most important species of the genus
Morus [1].This is native to Iran and belongs to both cultivated and wild mulberry varieties [2].The fruit is in
blackberry form and typically black, but sometimes dark blue with a sweet taste [3], and has been used as part of
traditional Chinese medicine for a long time [4], because the fruit of M. nigra is rich in compounds phenolics [5],
anthocyanins, proteins, and vitamins for urinary incontinence, depression, fever, cancer and diabetes [6]. Among the
phenolic compounds it has are gallic acid, ascorbic acid, p-coumaric acid, caffeic acid, to mention some have a great
nutritional and organoleptic significance and give the commercial characteristics of the fruits [7].
However, it is difficult to preserve fresh blackberry fruit due to its low acidity. In addition, phenolic compounds
are unstable in various solutions and, therefore, it is necessary to coat them to stabilize them, which can be achieved
by an encapsulation process [8]. For this reason, there is a real need to apply technologies to improve their useful
life, qualities nutritional, organoleptic and health benefits of blackberry fruit to boost commercial production with
economic and health benefits [9]. Encapsulation provides a means to control stability, solubility and bioavailability,
as well as for the release of bioactive components [10].
On the other hand, stability is the ability to verify the quality of a drug within its specifications. Stability tests
must be conducted under conditions that allow information on the stability of the product to be provided in the
shortest possible time, for which, the samples must be stored in conditions that accelerate the possible changes that
may occur during the validity period; Accelerated stability studies are carried out under exaggerated storage
conditions, to increase the rate of chemical, biological degradation or physical changes of a drug [11]. However,
there are not yet any studies that show the pharmaceutical stability of freeze-dried capsules of the fruit. M. nigra
from the Comarca Lagunera region. Therefore, the purpose of this study was to evaluate and investigate for the first