Agrawal et al Journal of Drug Delivery & Therapeutics. 2020; 10(5-s):224-228
ISSN: 2250-1177 [224] CODEN (USA): JDDTAO
Available online on 15.10.2020 at http://jddtonline.info
Journal of Drug Delivery and Therapeutics
Open Access to Pharmaceutical and Medical Research
© 2011-18, publisher and licensee JDDT, This is an Open Access article which permits
unrestricted non-commercial use, provided the original work is properly cited
Open Access Review Article
Solid Lipid Nanoparticle for the Delivery of Docetaxel: A Review
Agrawal Pranav*, Tatode Amol, Umekar Milind
Smt. Kishroitai Bhoyar College of Pharmacy, Department of Pharmaceutics, Kamptee, Nagpur, Maharashtra, India-441002
ABSTRACT
Solid lipid nanoparticles are the forefront of the rapidly developing field of nanotechnology with several potential applications in drug delivery,
clinical medicine and research. Due to its solid state it has greater stability than other nanocarrier systems. There are several other advantages
like sustained release, improves bioavaibility and delivery of poorly water soluble drugs, helps in control of several pharmacokinetic
parameters of drugs due to which use of SLN is increasing day by day. Various techniques can be used for the formulation of SLN i.e. solvent
evaporation, microemulsification technique, high pressure homogenization and supercritical fluid method. It has several applications likes it is
use in gene transfer therapy, also use in different drug delivery systmer like oral and pulmonary drug delivery system. Due to several
advantages SLNs are widely used in chemotherapy for the treatment of the cancer. The use of SLN for the delivery of Docetaxel to tumor site
have several benefits likes site specific delivery, less toxic effect, more cell cytotoxicity and more bioavaibility which leads to decrease in the
dosing frequency. Docetaxel is an anticancer agent extracted from plant Taxus Baccata which is widely used in chemotherapy to treat cancer.
This article contains the detail information of about the advantages, disadvantages, different method of preparation and several SLN loaded
with Docetaxel.
Keywords: Solid lipid nanoparticles, drug delivery, clinical medicine, poorly water soluble drugs
Article Info: Received 10 Aug 2020; Review Completed 15 Sep 2020; Accepted 23 Sep 2020; Available online 15 Oct 2020
Cite this article as:
Agrawal P, Tatode A, Umekar M, Solid Lipid Nanoparticle for the Delivery of Docetaxel: A Review, Journal of Drug Delivery
and Therapeutics. 2020; 10(5-s):224-228 http://dx.doi.org/10.22270/jddt.v10i5-s.4441
*Address for Correspondence:
Agrawal Pranav, Smt. Kishroitai Bhoyar College of Pharmacy, Department of Pharmaceutics, Kamptee, Nagpur,
Maharashtra, India-441002
Introduction
Colloidal particles ranging in size between 10 and 1000nm
are known as nanoparticles. They are manufactured from
synthetic or natural polymers and ideally suited to
optimized drug delivery and reduce toxicity. Over the years,
they have emerged as a variable substitute to liposome as
drug carrier. The successful implementation of nanopartilces
for drug delivery depends on their ability to penetrate
across the cell membrane, sustained release of their contents
and their stability
1
. There are several disadvantages of
liposome or traditional nanoparticles like stability, leakage
of drug from the dosage form, etc. to overcome these
problem Solid lipid nanoparticles was developed. SLN are
colloidal carriers developed in the last decade as an
alternative system to existing traditional carrier such as
emulsion, liposomes and polymeric nanoparticles. They are
a new generation of submicron-sized lipid emulsion where
the liquid lipid has been substituted by solid lipid. SLN offer
unique properties such as small size, large surface area, high
dose loading and the interaction of phases at the interfaces
and are attractive for potential to improve performance of
pharmaceuticals, neutraceuticals and other materials as well
as increase stability is the most important advantage of SLN.
SLN are sub-micron colloidal carrier which is composed of
physiological lipid, dispersed in water or in an aqueous
surfactant solution. The use solid lipid instead of liquid lipid
is beneficial as it has been shown to increase control over
the release kinetics of encapsulated compounds and to
improve the stability of incorporated chemically-sensitive
lipophilic ingredients. The benefit of using solid lipids is due
to several physiochemical properties of lipid. Firstly, the
mobility of reactive agents in solid matrix is lower than in a
liquid matrix and so the rate of chemical degradation
reactions may be retarded. Secondly, micro phase
separations of the active ingredients and carrier lipid within
individual liquid particles can be controlled, thereby
preventing the accumulation of active compounds at the
surface of lipid particles where chemical degradation
reactions often occur. There is also another benefit; the
absorption of poorly absorbed drugs has been shown to be
increased after incorporation into solid lipid nanoparticles
2
.
Due to several benefits SLN are used for various types of
drugs like antineoplastic agents, delivery of several protein
and peptide, antiepileptic agents, etc. Cancer is one of the