Synthesis and oxidation study of the simplest binuclear metallocene compound of osmium, biosmocene Hiroki Yasuhara, Kazuki Koga, Satoru Nakashima * Department of Chemistry, Graduate School of Science, Hiroshima University, Kagamiyama, Higashi-Hiroshima 739-8526, Japan article info Article history: Received 21 October 2014 Received in revised form 20 December 2014 Accepted 22 December 2014 Available online 27 December 2014 Keywords: Biosmocene Mixed-valence state Variable-temperature NMR Valence-detrapping abstract Selective mono-lithiation method of bis(cyclopentadienyl)osmium(II) (osmocene) was established. Iodoosmocene(C 5 H 4 I)Os(C 5 H 5 ) (OcI), which is the rst monohalogenated product of osmocene, was prepared by the reaction of lithioosmocene with I 2 . Ullmann coupling reaction of iodoosmoene allowed to prepare biosmocene(C 5 H 5 )Os(m 2 -h 5 :h 5 -C 10 H 8 )Os(C 5 H 5 ) (OcOc). OcOc reacted with I 2 , giving mixed- valence biosmocenium salt [(C 5 H 5 )Os II (m 2 -h 5 :h 5 -C 10 H 8 ) (C 5 H 5 )Os IV I]I 3 (A). The structure of A was deter- mined by single crystal X-ray structural analysis. The intramolecular electron transfer reaction between Os II and Os IV was observed by using 1 H NMR spectroscopy, accompanied by the exchange of I anion between the two units. The activation energy of the electron transfer reaction was estimated and the value was larger than that of binuclear ruthenocenium salt [(C 5 H 5 )Ru II (m 2 -h 5 :h 5 -C 10 H 8 ) (C 5 H 5 )Ru IV I]I 3 (B). © 2015 Elsevier B.V. All rights reserved. Introduction There have been many investigations concerning the mixed valence state of binuclear metallocene derivatives of iron [1e6] and ruthenium [7e10], while such study about osmium derivative has not been reported. Any attempts for synthesis of the simplest binuclear metallocene compound of osmium, namely biosmocene (OcOc), resulted in failure [8,11], and even monohalogenated osmocene compound, which is considered as useful precursor of binuclear compounds, had not been prepared. Although prepara- tion method of decahalogenated osmocene derivatives (C 5 X 5 ) 2 Os(X ¼ Cl, Br, I) has been reported [12], these halides are obviously inconvenient for synthetic experiment because of the poor solubility, preparation difculty and need of toxic mercury reagent for preparation. First of all, we had to nd the facile and useful halogenation method of osmocene for development of the binuclear osmocene chemistry. As for ferrocene and ruthenocene, R. Sanders and U. T. Muller-Westerhoff established the selective mono-lithiation method of these methallocens [13], and M. S. Inkpen et al. reported that mono-iodoferrocene (C 5 H 4 I)Fe(C 5 H 5 ) (FcI) was isolated by the reaction of mono-lithioferrocene (C 5 H 4 Li) Fe(C 5 H 5 ) (FcLi) and I 2 [14]. Using this synthesis strategy, we succeeded in selective preparation of mono-iodoosmocene(OcI) in 77% yield. OcI is the rst example of monohalogenated product of osmocene. In general, Ullmann coupling reaction readily generates biaryl compound from two aryl iodides. Therefore, we selected this type of reaction for preparation of OcOc. The attempt was suc- cessful, and OcOc was obtained in moderate yield (48%). It was reported that mixed-valence biruthenocenium salt [(C 5 H 5 )Ru II (m 2 -h 5 :h 5 -C 10 H 8 ) (C 5 H 5 )Ru IV I]I 3 (B) [8] was generated by oxidation of RcRc with two equivalent mol of I 2 . Intramolecular electron transfer reaction between two Ru centers was observed for a solution of B by using 1 H NMR spectroscopy. For the observation of the similar reaction between two Os centers, we attempted oxidation of OcOc by I 2 , then succeeded in isolation of mixed- valence biosmocenium salt [(C 5 H 5 )Os II (m 2 -h 5 :h 5 -C 10 H 8 ) (C 5 H 5 ) Os IV I]I 3 (A). A was characterized by 1 H NMR, ESI-MS and elemental analysis, and the structure was determined by single-crystal X-ray structural analysis. Intramolecular electron transfer reaction of A was also observed by variable-temperature 1 H NMR measurement. Herein, we discuss the synthesis and oxidation state of OcOc by comparing them with the corresponding Ru analogs. Experimental General information All reactions were performed under an argon atmosphere unless explicitly mentioned, while purication procedure was carried out * Corresponding author. Natural Science Center for Basic Research and Devel- opment (N-BARD), Hiroshima University, Kagamiyama, Higashi-Hiroshima 739- 8526, Japan. Tel.: þ81 82 424 6291. E-mail address: snaka@hiroshima-u.ac.jp (S. Nakashima). Contents lists available at ScienceDirect Journal of Organometallic Chemistry journal homepage: www.elsevier.com/locate/jorganchem http://dx.doi.org/10.1016/j.jorganchem.2014.12.030 0022-328X/© 2015 Elsevier B.V. All rights reserved. Journal of Organometallic Chemistry 779 (2015) 86e90