J. Acad. Indus. Res. Vol. 1(5) October 2012 281
©Youth Education and Research Trust (YERT) Nomila Merlin et al., 2012
ISSN: 2278-5213
Taxol production by endophytic Fusarium solani LCPANCF01 from Tylophora indica
J. Nomila Merlin
1
, I.V.S. Nimal Christhudas
2
, P. Praveen Kumar
2
, M. Kumar
3
and P. Agastian
2
1
Dept.of Biotechnology, Bharathiar University, Coimbatore-641046, TN, India
2
Dept. of Plant Biology and Biotechnology, Loyola College, Chennai-600034, TN, India
3
Dept. of Plant Biology and Plant Biotechnology, Madras Christian College, Tambaram, Chennai-600059, TN, India
agastian@loyolacollege.edu; +91 9444433117
_____________________________________________________________________________________________
Abstract
Twenty five endophytic fungal isolates were obtained from the roots of Tylophora indica (Burm. f) and
screened for the presence of an anticancer drug, taxol. Among the 25 isolates, Fusarium solani LCPANCF01
was identified based on the micro morphology, cultural characteristics and sequence analysis using internal
transcribed spacer (ITS1 and ITS4). Fusarium solani LCPANCF01 strain was grown in M1D liquid medium
for 21 d and extracted with dichloromethane. The presence of taxol was confirmed by TLC, HPLC, UV, IR,
and ESI-MS spectroscopy analysis by comparing with the standard drug.
Keywords: Tylophora indica, Fusarium solani, dichloromethane, taxol, anticancer drug.
Introduction
Taxol is isolated from the barks of pacific yew tree
(Taxus brevifolia) (George et al., 1994; Dewick, 2009)
and the most important antimitotic agent which is active
against lung, ovarian, breast, head-neck cancer and
advanced forms of Kaposi's sarcoma. Taxol inhibits cell
proliferation by binding to the β-subunit of the tubulin
heterodimers, thus promoting its polymerization (Kovacs
et al., 2007). However, a complete course of treatment
per patient may requires 2 g of taxol administered
several times over many months. To obtain 1 kg of taxol,
it requires 3000 yew trees (10,000 kg of bark) and
current demand of taxol is 250 kg per annum (Dewick,
2009). This insufficiency of taxol and environmental issue
of harvesting from trees demands researcher to discover
the alternate technique for the production of taxol.
Taxol is now obtained by several methods, e.g. total
chemical synthesis (Nicolaou et al., 1994),
semi-synthesis from its precursor (Commercn et al.,
1995), plant tissue or cell culture (Hu et al., 2003).
Endophytic fungus from various taxus species produces
taxol although the amounts are very small. First taxol
producing endophytic fungi T. andreanae is from Taxus
brevifolia (Stierle et al., 1993). Since then, many other
endophytic fungi from other plant species have been
successfully reported to produce taxol (Strobel et al.,
1996; Li et al., 1996). Tylophora indica (Burm. f)
(Asclepiadaceae) is a climbing perennial plant that grows
in India, commonly called as antmool in Ayurveda. The
leaves of Tylophora have been traditionally used as a
folk medicine. It has been used for respiratory problems
such as asthma, allergies, bronchitis and common cold.
The roots and leaves contain 0.2 to 0.46% of
therapeutically important alkaloids namely tylophorine,
tylophorinine and tylophrinidine.
Major alkaloid tylophorine has immunosuppressive,
anti-inflammatory (Gopalakrishnan et al., 1979),
anti-tumor (Donaldson et al., 1968) and anti-amoebic
(Bhutani et al., 1987) properties. Since, T. indica is an
endemic plant an attempt is made to conserve the
medicinal plant through exploration of endophytic fungi
and screened for its taxol production.
Materials and methods
Plant collection: Tylophora indica fresh plants were
collected from Kerala Forest Research Institute (KFRI),
Trissur, Kerala, South India during the month of January
2012 (Fig. 1). The taxonomical identity of the plant was
confirmed by Dr. D. Narashiman, Department of Botany,
Madras Christian College, Tambaram, South India.
Fig 1. Tylophora indica.
RESEARCH ARTICLE