Liposome and Polysaccharide Based Nanomedicines: An Emerging Hope
to Improve the Peritoneal Dialysis Technique
Guleria A and Kumar D
*
Centre of Biomedical Research (CBMR), Lucknow-226014, Uttar Pradesh, India
*
Corresponding author: Kumar D, Centre of Biomedical Research (CBMR), SGPGIMS Campus, Raibareli Road, Lucknow-226014, Uttar Pradesh, India, Tel:
+91-8953261506, 8005409932; E-mail: dineshcbmr@gmail.com
Received date: November 03, 2016; Accepted date: December 08, 2016; Published date: December 12, 2016
Copyright: © 2016 Guleria A, et al. This is an open-access article distributed under the terms of the Creative Commons Attribution License, which permits unrestricted
use, distribution, and reproduction in any medium, provided the original author and source are credited.
Keywords: Polysaccharide based Nanoparticles; Antimicrobial
nanomaterials; Biological synthesis; Peritoneal dialysis; Renal
replacement therapy; Health care infections; Infectious peristonitis
Introduction
Peritoneal Dialysis (PD) is the simple and cost-efective renal
replacement modality used for treating patients with End-Stage Renal
Failure (ESRF) [1-3]. It ofers several clear advantages over
Hemodialysis (HD) like cost-efectiveness, fexibility and autonomy to
the patients, however, it is ofen associated with a high risk of infection
of the peritoneal cavity, subcutaneous tunnel and catheter exit site as
well as the subsequently formed microbial bioflms. In current practice,
the episodes of PD associated infections-if diagnosed timely-are cured
through the empirical use of antibiotics. However, the fungal infections
or infections caused by drug resistant bacteria remains critical and
ofen lead to infammation of the peritoneum. Te complication-
generally known as infectious peritonitis-is not only the major cause of
technique failure and patient transferring to HD, it is also the leading
cause of mortality and morbidity in ESRF patients continuing on PD.
As the number of ESRF patients continuing on PD is increasing
continuously every year, the PD associated infections are also
becoming more and more evident posing extra burden on dialysis-
centers/nephrology-wards to resolve such life-threatening and critical
conditions. Te situation is even more pathetic and worse in
developing countries-having limited healthcare centers and poor
socioeconomic status of patients-where majority of ESRF patients
continuing on PD die because of intraperitoneal (IP) infections [1,3-5].
As ESRF patients are generally manifested with sabotaged immune
system, therefore, high antibiotic dose is ofen used to achieve
complete eradication of Intraperitoneal (IP) infections. However, the
frequent intraperitoneal administration of higher anti-biotic doses may
cause serious side-efects including peritoneal malfunctioning and
hepatotoxicity. Tus, there has been an urgent need to improve the PD
technique in terms of reducing the frequency of IP infections and
improving its efciency to remove drugs/endotoxins from the patient
body.
Nanomedicines
Tere are several reports in the literature now where
nanotechnology products including nanomedicines have been
implicated in the diagnosis and treatment of kidney diseases [6]. Tere
is also an increasing cohort of nanomaterials which has been envisaged
to improve the PD technique either through the use of (a) anti-
microbial spray for preventing Catheter Exit-Site Infection [7], (b)
liposomes for detoxifcation of drugs and endogenous metabolites to
enhance the efciency of peritoneal dialysis [8,9], (c) nano-carriers for
TNF-β1-SiRNA to inhibit the peritoneal fbrosis [10], (d) silica-
containing redox nanoparticles (siRNPs) for high-performance
peritoneal dialysis through suppressing oxidative stress by scavenging
Reactive Oxygen Species [11], and (e) antimicrobial nanomaterials
synthesized biologically–which confer several advantages like
biocompatibility, low cellular toxicity and activity against variety of
drug-resistant bacteria- to impart infection resistant properties to the
PD fuid and thus reducing the frequency of PD associated infections
[12]. An alternative, but more relevant and promising approach to
improve the existing PD therapy-in terms of its dialysis efciency and
limiting microbial infections- can be envisaged based on the use of
liposomal antibiotic formulations [13,14]. Liposomes-generally
referred as nanometric size vesicles formed by phospholipid bilayer
membrane-exhibit remarkable physicochemical properties like
biocompatibility, biodegradability, and low cytotoxicity. On top of this,
these (a) may increase the solubility of hydrophilic, hydrophobic and
amphiphilic molecules of therapeutic potential, (b) may protect them
from degradation in the body and (c) may enhance their retention
time within the peritoneal cavity [13-16]. All these features are highly
desirable for increasing dialysis efciency and treatment against of
formidable intraperitoneal infections in PD patients. Terefore, we
strongly believe that liposomal formulations will soon enter into the
peritoneal dialysis therapy: (a) to reduce the in vivo toxicity of anti-
biotics for their safe intraperitoneal use and/or (b) to improve the
therapeutic efcacy of poorly water soluble antibiotics [13,16].
Similarly, the nanometric drug-delivery systems derived from natural
polysaccharides -such as heparin, cellulose, chitin, chitosan,
cyclodextrin, dextrose, etc. can also be envisaged for efective and
complete eradication of IP infections [17-22]. Natural polysaccharides
represent a novel class of permeative biopolymers and because of their
stability, availability, renewability, low toxicity and low cost are gaining
tremendous popularity in the development of nano-sized drug delivery
systems [23]. Various functional groups such as hydroxyl, amine etc.
which are present in these polysaccharides allows chemical
derivatization by which their properties can be modulated and
adjusted to the aimed application [23-25]. Tese are the reasons that
polysaccharides based biomaterials have undergone rapid development
in the past few decades for their use in a variety of biomedical and
pharmaceutical applications such as drug delivery (or co-delivery of
synergistic drug combinations), gene therapy, vascular grafs, and
scafolds for tissue engineering, wound dressings, medical implants
and medical imaging [17,22]. In the context of improving PD
technique, we foresee a great potential of low molecular weight heparin
based nano-sized drug delivery systems. Heparin-most commonly
known as an anticoagulant-is commonly administered
intraperitoneally whenever fbrin is detected in the dialysate efuent (a
clinical manifestation of peritonitis) [26]. A variety of recent research
studies have shown that heparin improves the biocompatibility of
Guleria and Kumar, Pharm Anal Acta 2016, 7:12
DOI: 10.4172/2153-2435.1000524
Commentry Open Access
Pharm Anal Acta, an open access journal
ISSN: 2153-2435
Volume 7 • Issue 12 • 1000524
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ISSN: 2153-2435
Pharmaceutica Analytica Acta