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Magnano, et al: TNF in hand OA
Personal non-commercial use only. The Journal of Rheumatology Copyright © 2007. All rights reserved.
A Pilot Study of Tumor Necrosis Factor Inhibition in
Erosive/Inflammatory Osteoarthritis of the Hands
MOLLYD.MAGNANO,ELIZAF.CHAKRAVARTY,CORRIEBROUDY,LORINDACHUNG,ARIELLAKELMAN,
JENNIFERHILLYGUS,andMARKC.GENOVESE
ABSTRACT. Objective. To determine if anti-tumor necrosis factor (TNF) therapy (adalimumab) can safely improve
symptoms of erosive/inflammatory osteoarthritis (EOA).
Methods. Thiswasanopen-labelpilottrialin12patientswithEOA.Patients>45yearsoldwithEOA
of the hands defined by ≥ 2 tender and ≥ 2 swollen joints (distal interphalangeal, proximal interpha-
langeal, first carpometacarpal) despite nonsteroidal antiinflammatory drug therapy were eligible.
Patientswereexcludedforautoimmunearthritis,recentdiseasemodifyingantirheumaticdruguse,prior
use of anti-TNF therapy, infection, malignancy, or poorly controlled medical conditions.All patients
receivedadalimumab40mgeveryotherweekfor12weeks.Safetywasassessed4weeksafterthefinal
dose. Primary endpoints included safety andAmerican College of Rheumatology (ACR) response.
Results. Patientswerepredominantlyfemalewithameanageof60yearsand12yearsofarthritis.All
patients completed the study and safety followup.Adverse events were mild without necessitating dis-
continuation of study drug. After 12 weeks, there was a statistically significant improvement in the
number of swollen joints compared to baseline (p < 0.01). One patient achieved an ACR20 response
and 42% achieved an OMERACT-OARSI response.Although we detected no statistically significant
improvement in the number of tender joints, grip strength, disability, pain, or global disease assess-
ments, trends suggested modest improvement in all efficacy measures.
Conclusion. Thissmallopen-labelstudyofpatientswithEOAdemonstratedthatadalimumabwaswell
tolerated. Treatment with adalimumab for 3 months did not significantly improve the signs and symp-
toms of EOA and most patients did not achieve an ACR20. Trends suggested improvement and indi-
vidualpatientshadsomebenefit.Factorslimitinginterpretationofthisstudyincludethelackofacon-
trol group, outcomes chosen, number of patients treated, and the duration of treatment. (First Release
May 15 2007; J Rheumatol 2007;34:1323–7)
Key Indexing Terms:
OSTEOARTHRITIS TUMORNECROSISFACTOR TREATMENT CYTOKINE
From the Division of Immunology and Rheumatology, Stanford University,
Palo Alto, California, USA.
Supported by Abbott Pharmaceuticals and grant 5 M01 RR000070 from
the National Center for Research Resources, National Institutes of Health.
M.D. Magnano, MD, Postdoctoral Fellow; E.F. Chakravarty, MD,
Assistant Professor; C. Broudy, MD, Postdoctoral Fellow; L. Chung, MD,
Assistant Professor; A. Kelman, MD, Adjunct Clinical Professor, Stanford
University, Medical Director, Genentech Inc.; J. Hillygus, Research
Assistant; M. Genovese, Associate Professor of Medicine, Division of
Immunology and Rheumatology, Stanford University.
Address reprint requests to Dr. M. Genovese, Division of Immunology and
Rheumatology, Stanford University, 1000 Welch Road, Suite 203, Palo
Alto, CA 94304. E-mail: genovese@stanford.edu
Accepted for publication February 26, 2007.
Osteoarthritis (OA) is a heterogeneous group of conditions
with defective integrity of articular cartilage and changes in
underlyingbone.ThepathogenesisofOAismultifactorialand
involves a complex interplay of genetic, metabolic, biochem-
ical, and biomechanical factors with variable components of
inflammation. A subset of patients with OA develop an
inflammatory and erosive form of the disease. Erosive
osteoarthritis (EOA) is clinically recognized in peri-
menopausalfemalepatientswhodevelopsynovitisinthedis-
tal and proximal interphalangeal (DIP, PIP) joints of the
hands.TheclassicradiologicalchangesofEOAarecharacter-
ized by a combination of bony proliferation and central ero-
sionsresultingintheclassic“gull-wingdeformity.”Inclinical
studies, the diagnosis of EOA is accepted only for patients
meeting American College of Rheumatology (ACR) clinical
criteria for OA of the hand and showing radiographic aspects
of articular surface erosions
1
.
Agrowingbodyofevidencesupportsthetheorythataber-
rant cytokine biology is important to the pathophysiology of
OA.MorphologicalchangesobservedinOAincludecartilage
erosion as well as variable degrees of synovial inflammation.
Cartilagefromequineosteoarthritickneesdemonstrateslevels
of interleukin 1ß (IL-1ß), tumor necrosis factor-α (TNF-α),
and numerous matrix metalloproteinases (MMP) above those
foundinnormaljoints
2
.Thiscytokinemilieusignalssynovio-
cytes and chondrocytes to express metalloproteinases that
destroy the structural integrity of synovial cartilage
3
. In
response to this inflammatory environment, chondrocytes
show a diminished capacity to self-repair in response to
growth factors, resulting in irreversible cartilage damage
4
.
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