www.ijbcp.com International Journal of Basic and Clinical Pharmacology | November-December 2016 | Vol 5 | Issue 6 Page 2352
IJBCP International Journal of Basic and Clinical Pharmacology
Print ISSN: 2319-2003 | Online ISSN: 2279-0780
Original Research Article
Pentobarbitone-induced sleeping time and sub-acute toxicity studies of
Trichilia monadelpha aqueous extract
George Owusu
1,3
, Meshack Antwi-Adjei
2,3
, Isaac T. Henneh
2,3
*
INTRODUCTION
Trichilia monadelpha (Thonn) JJ De Wilde (fam.
Meliaceae) is a medium-sized tree that grows up to 20m
high in the tropical rain forest in West Africa. Different
parts of the plant are used either alone or in combination
with other plants for treatment of many diseases in West
Africa.
1
Previously, the inhibitory effects of the aqueous, hydro-
ethanol and petroleum ether extracts of the stem bark of
the plant in carrageenan-induced paw oedema in 7-day-
old chicks and Complete Fruend’s adjuvant-induced
arthritis in rats has been reported.
2
Also, the analgesic
effect of the hydro-ethanol, petroleum ether and ethyl
acetate extracts of the stem bark of the plant has been
earlier reported.
3
Again, the antioxidant potential and
phytochemical constituents of the stem bark extracts of
the plant have been evaluated.
4
Moreover, the plant has
been reported to possess antiplasmodial and
antitrypanosomal properties.
5
Despite the numerous
activities of the plant reported in literature, there is no
valid scientific data on its hypno-sedative effects and
toxicity profile.
ABSTRACT
Background: Trichilia monadelpha is used either alone or in combination with
other plants to treat many diseases in West Africa. Earlier, the anti-
inflammatory, analgesic and anti-parasitic effects of the plant have been
investigated to confirm its folkloric use. The current study is aimed at
investigating the sub-acute toxicity profile as well as hypno-sedative effect of
the Trichilia monadelpha aqueous extract (TAE).
Methods: For the pentobarbitone-induced sleeping test, rats (150-200 g, n=5)
were pre-treated with TAE (100, 300 and 1000 mg/kg, p.o.) or distilled water
(control group) 30 minutes before they were challenged with Pentobarbitone
Sodium (50 mg/kg body weight, i.p). Sleeping time of each animal was
recorded and analysed. In the sub-acute toxicity test, rats were treated daily
either TAE (30, 100 and 1000 mg/kg) or water (control group) for two weeks
after which the animals were sacrificed. Blood samples were collected for
haematological and biochemical analyses. Specific organs were then removed
and weighed immediately.
Results: The pentobarbitone-induced sleeping test resulted in a significant and
dose-dependent increase in the duration of sleep of the rats. There were
however no significant changes in the relative weight of vital organs of the
control and TAE treated groups. Similarly, there were no significant differences
in haematological and biochemical parameters between control and TAE treated
groups.
Conclusions: TAE significantly and dose-dependently increased the duration of
pentobarbitone-induced sleeping time in rats. TAE showed no significant
changes in the relative weight of the vital organs, haematological and
biochemical parameters.
Keywords: Trichilia monadelpha, Pentobarbitone, Hypno-sedative, Sub-acute
toxicity
DOI: http://dx.doi.org/10.18203/2319-2003.ijbcp20164088
1
Department of Pharmacology,
School of Medicine, University
for Development Studies,
Tamale, Ghana
2
Department of Pharmacology,
School of Medical Science,
University for Development
Studies, Tamale, Ghana
3
Department of Pharmacology, ,
Faculty of Pharmacy and
Pharmaceutical Sciences,
Kwame Nkrumah University of
Science and Technology,
Kumasi, Ghana
Received: 20 September 2016
Accepted: 20 October 2016
*Correspondence to:
Mr. Isaac T. Henneh,
Email: i.t.henneh@
uccsms.edu.gh
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