American Journal of Medicine and Medical Sciences 2019, 9(10): 396-400
DOI: 10.5923/j.ajmms.20190910.09
Research of Polymorfic Locus (430 C/T) of CYP2c9/*2
Gene Distribution Frequencies among Patients with
Epilepsy
Nodira Miratalievna Tuychibaeva
1,*
, Parakhat Rustamovna Alimkhodzhaeva
1
,
Kodirjon Tuhtabaevich Boboev
2
1
Department of Nervous Diseases, Tashkent Medical Academy, Tashkent, Uzbekistan
2
Department of Molecular Medicine and Cell Technologies, Scientific Research Institute of Hematology and
Blood Transfusion of the Ministry of Health of the Republic of Uzbekistan, Tashkent, Uzbekistan
Abstract The aim of the study was to establish the association of polymorphism (430 C/T) of the CYP2C9/*2 gene with
the risk of developing pharmacoresistant epilepsy. The study included patients with pharmacoresistant and controlled forms
of epilepsy. There was a tendency to associate the T allele and the heterozygous C/T genotype with the pharmacoresistant
form of epilepsy.
Keywords Polymorphism (430 C/T), CYP2C9/*2 gene, Pharmacoresistant epilepsy, Allele, Genotype
1. Introduction
The problem of treating a pharmacoresistant form of
epilepsy is the subject of a study by various authors [4a],
but so far an effective method of treatment and prediction of
this pathology has not been found. The basis of the
treatment of epilepsy is a long-term lifelong intake of
antiepileptic drugs [3]. The criterion of effective
antiepileptic therapy can be considered the complete
absence or minimization of side effects and complications
of therapy [1,2,12,13].
One of the most effective ways to improve drug therapy
is a personalized approach to treatment, requiring the study
of the molecular genetic basis of the disease. As you know,
one of the key roles in drug metabolism is played by
cytochrome P450 [6,11,14,18,17]. In this regard, the study
of the cytochrome P450 2C9 gene (CYP2C9) is of
considerable interest to researchers, in which polymorphic
changes are attributed to the development of undesirable
complications against the background of pharmacotherapy
for epilepsy and, inter alia, when taking valproic acid
[8,5,9,10,15,19,21].
In this regard, the study of one of the poorly studied
polymorphisms (430 C/T) of the CYP2C9/*2 gene is of
* Corresponding author:
alteam2201@gmail.com (Nodira Miratalievna Tuychibaeva)
Published online at http://journal.sapub.org/ajmms
Copyright © 2019 The Author(s). Published by Scientific & Academic Publishing
This work is licensed under the Creative Commons Attribution International
License (CC BY). http://creativecommons.org/licenses/by/4.0/
interest for studying the etiopathogenetic basis of
pharmacoresistant epilepsy [7].
2. Main Body
2.1. The Purpose of Our Research
The purpose of this study was to establish the association
of polymorphism (430 C/T) of the CYP2C9/*2 gene and the
risk of developing pharmacoresistant epilepsy.
2.2. Material and Methods of Study
The study included a total of 382 subjects, including the
main group consisting of 124 people, including 77 patients
with pharmacoresistant epilepsy (1a-subgroup) and 47
patients with controlled epilepsy (1b-subgroup). The control
group consisted of 134 healthy individuals.
The diagnosis was established on the basis of clinical and
anamnestic examination and laboratory studies. In patients
with an established diagnosis in the main group and
conditionally healthy individuals in the control group, a
study was made of the distribution of polymorphic locus
(430 C/T) in the CYP2C9/*2 gene.
DNA was isolated from venous blood using a DNA sorb
and “Ribo-Sorb” kit (AmpliSens®, Russia). The
concentration and purity of the isolated DNA was
determined on a NanoDrop 2000 instrument (USA).
Genotyping of polymorphism (430 C/T) in the
CYP2C9/*2 gene was performed by PCR-RFLP using an
Applied Biosystems 2720 instrument.