Brain Research, 201 (1980) 129-141 129
© Elsevier/North-Holland Biomedical Press
A STUDY OF THE QUANTAL (ALL-OR-NONE) CHANGE IN REFLEX
LATENCY PRODUCED BY OPIATE ANALGESICS
JON D. LEVINE*, DENNIS T. MURPHY, DAVID SEIDENWURM, ANNE CORTEZ and
HOWARD L. FIELDS
Departments of Neurology and Physiology, University of California, San Francisco, Calif. 94143
( u.s.,4.)
(Accepted June 5th, 1980)
Key words: pain -- opiates -- reflexes-- analgesia
SUMMARY
The properties of opiate-induced changes of tail-flick latency were studied in the
rat.
(1) Morphine and pentazocine produced a stepwise increase in latency which
rose from near baseline to cut-off (usually greater than 20 see) in less than 30 sec.
Abrupt return to pre-treatment latencies was observed either spontaneously or when
the rat was back-titrated with the narcotic antagonist naloxone.
(2) The proportion of rats showing this stepwise change increased with in-
creasing dose; however, the step itself was independent of dose. The same step was
produced by a slow, constant infusion of morphine but was not produced by ice-water
stress or barbiturate administration.
(3) Increasing heat intensity to the tail shortened the baseline latency and raised
the mean dose of morphine required to produce a step latency increase.
(4) A step increase in latency was also observed when paw withdrawal instead of
tail-fl{ck was measured.
We hypothesize that the analgesic behavior described partly defines the oper-
ating characterisitics of art intrinsic endorphin-mediated analgesia system which
mediates narcotic suppression of withdrawal reflexes.
INTRODUCTION
Opiates are the most potent analgesic agents presently in use. Great progress has
* To whom all correspondence is to be addressed at the Department of Neurology.