Pal et al Journal of Drug Delivery & Therapeutics; 2014, 4(2), 47-51 47
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RESEARCH ARTICLE
FORMULATION AND EVALUATION OF NUTRACEUTICAL TABLET USING
HERBAL DRUGS BY DIRECT COMPRESSION METHOD
Upendra Nagaich
1
, *Ashok Kumar Pal
2
, Charu Bharti
2
, Neha Gulati
2
1
Department of Pharmaceutics, Amity Institute of Pharmacy, Amity University, Noida [Uttar Pradesh] India
2
Department of Pharmaceutics, School of Pharmacy, Bharat Institute of Technology, Partapur By Pass Road, Meerut-
250103 [Uttar Pradesh]
*Corresponding Author’s Email: apal11595@gmail.com , 08791575261
INTRODUCTION
Oral route has been one of the most popular routes of
drug delivery due to its ease of administration, patience
compliance, least sterility constraints and flexible design
of dosage forms.Tablets are defined as unit dose, temper
evident solid preparations containing one or more active
ingredients. Conventional drug delivery systems like
tablets and capsules often dissolve rapidly in the
gastrointestinal tract for absorption into the bloodstream
give rise to inordinately high drug concentrations in
plasma
1
. The concept of making utility of food as health
promoting factor beyond its nutritional value is gaining
acceptance with in public arena and among scientific
community. Nutraceuticals contain health- supporting
ingredients or natural components that have an ability
health benefit for the body.
2
A „nutraceutical‟ is a
product isolated or purified from foods that is generally
sold in medicinal forms not usually connected with food.
A nutraceutical is bearing to have a physiological benefit
or give protection against chronic disease. Term coined
by Dr. Stephen L De Felice, Founder and Chairman of
the Foundation for Innovation in Medicine, New Jersey,
USA. Nutraceuticals sometimes referred as “functional
foods”, have caused heated debate because they change
the traditional dividing line between food, and medicine.
3
A nutraceutical is “any non-toxic food component that
has scientifically proven health benefits, including
disease treatment or prevention.” The functional
component of the food must be standardized in the
nutraceutical product and generate under good
manufacturing practices (GMPs).
4
Increased public
demand, trends in demography, socio-economic
scenario. More researches and studies, nearly two thirds
of the world‟s 6.1 billion people rely on the healing
power of plant based materials for many reasons-
availability, affordability, safety or their belief in
traditional affordability, safety or their belief in
traditional cures Medical benefits of food have been
investigated for thousands of years. Modern nutraceutical
industry began to develop in Japan during the 1980s.
Various benefits of nutraceuticals are may help us live
longer, may increase the health asses of our diet, help us
to abstain particular medical condition, it have a
psychological advantage from doing something for
oneself, and may be sensed to be more "natural" than
traditional medicine and less likely to produce unpleasant
side-effects.
3, 5
The nutraceuticals normally contains required amount of
lipids, protein, carbohydrates, vitamins, minerals and
other necessary nutrients depending upon their
emphases. Nutraceuticals in the market contains both
traditional foods and non-traditional. When a supplement
tablet is ingested, the body must digest and absorb the
nutrients. Nutraceutical may include a whole area of
products like isolated nutrients, dietary supplements,
herbal products and other processed foods.
5
The
growing disapproval among the patients about the
synthetic therapeutic agents and affect about their
toxicological profile gave birth to the “Dietary
Supplements Health and Education Act” (DSHEA) in
USA in 1994.
5, 6
The concept behind the mode of action
of nutraceutical dosage form is to provide functional
benefits by enhancing the supply of natural building
blocks. It works in to two ways that is to minimize
diseases sign or to improve body performance.
2, 3
Clove consists of dried flower buds of Eugenia
caryophyllus, family Myrtraceae. The cloves on drying
become perfectly crimson or brownish-black in colour.
Clove is used as a dental analgesic, carminative,
stimulant, flavouring agent an aromatic and antiseptic.
Cinnamon consist of dried inner bark of shoots of
coppiced trees of Cinnamon zeylancium Nees. Bark is
ABSTRACT
Aim: The objective of present study was to formulate and evaluate the nutraceutical tablets with different combination of
herbal drugs. Material and Method: The nutraceutical tablet containing lactose and mannitol as diluent and containing
natural drugs like clove and cinnamon which was prepared by direct compression method. The compressed formulations were
subject to several evaluation parameters like appearance, thickness, weight variation, hardness and friability. Results: The
results of all evaluation parameters of nutraceutical tablet were within the acceptable limit. Pre-compression studies of
nutraceutical tablet show satisfactory results. The thickness, hardness, weight variation, and friability of nutraceutical tablet
were found to in acceptable range. The in-vitro drug release of eugenol from optimised nutraceutical formulation was found to
be 90.23%. Significant results were obtained from present study. Discussion: The finding of current investigation clearly
found that the health promotion of the body could be done by nutraceuticals.
Keywords: Direct compression, Nutraceutical, Eugenol, In-vitro drug release.