Volume 1 • Issue 6 • 1000e130
Biochem Pharmacol
ISSN:2167-0501 BCPC, an open access journal
Editorial Open Access
Shah et al., Biochem Pharmacol 2012, 1:6
DOI: 10.4172/2167-0501.1000e130
Cancer afects a signifcant proportion of the population of the
United States and the rest of the world. In the U.S. approximately
12 million people were directly afected by cancer in 2010 [1]. In a
signifcant percentage of these patients, the disease will become invasive
and may eventually be the primary cause of death. Classical treatment
of cancer involves surgery, radiation and chemotherapy. However,
chemo and radiation therapies cause more harm rather than help in
the long run as it is becoming evident that radiation/chemo therapies
induce mutations that could transform the tumor into a drug-resistant
and metastatic cancer [2-4]. Recent advances in cancer biology provide
a hope for the development of novel, personalized and targeted therapy
for cancer patients. Among many new directions of research in cancer,
the understanding of the mechanisms that transform a localized tumor
into an invasive one is the most exciting.
Although cancer is frequently considered as a disease of abnormal
proliferation and accelerated abnormal growth, cancer progression
is not determined solely by proliferative advantage of malignant cells
within a tumor [5]. Other factors such as resistance to apoptosis and
ability to bypass senescence pathways also contribute signifcantly
to the process [6]. Correct adhesion between adjacent epithelial cells
is important in determining the normal structure and function of
epithelial tissues [7]. Accumulating evidence suggests that dysregulated
cell-cell adhesion is associated with development and progression of
most epithelial cancers [8].
Cell-cell adhesion is a critical component for the assembly of
coherent sheets of barrier-forming epithelial cells that eventually line
most organs, ducts and lobules. However, it is now understood that
cell-cell contacts are not static structures that maintain barriers by just
holding cells together. Tese contacts undergo constant remodeling to
allow extrusion of apoptotic cells and to replace them with newly formed
epithelial cells without the loss of barrier function. Cell-cell contacts
are also remodeled to meet special physiological and developmental
needs such as puberty, pregnancy, lactation, or involution. During
wound healing, epithelial cells undergo coordinated movement and
proliferation to bridge the wound, and establish new cell-cell contacts
with epithelial cells from the opposing side of the wound [9-11].
Epithelial cell-cell contacts consist of three main adhesive
structures: tight junctions (TJs), adherens junctions and desmosomes,
as well as gap junctions. In polarized epithelial cells the TJs and
adherens junctions are asymmetrically distributed at the apical region
of the lateral membrane. Tis asymmetry forms the apical junctional
complex, which encircles the apex of the cells and marks the border
between apical and basolateral membrane domains [9,12]. Tese
adhesive structures are composed of integral transmembrane proteins
such as claudins or occludin that link the neighboring cells through
homophilic and heterophilic interactions. Tese transmembrane
proteins are anchored to cytoskeleton by zonula occludens proteins,
which also organize signaling complexes and anchor cell-cell contacts
to the actin cytoskeleton [13,14]. Especially, zonula occludens-1
(ZO-1) plays a key role in organizing TJs by serving as a scafold and
providing multiple interaction domains where several transmembrane
and signaling proteins can bind to form the TJ structure [13,15,16].
As the most apical structure between epithelial and endothelial cells,
TJs control paracellular difusion of ions and certain molecules [17].
In addition, TJs play a vital role in maintaining cell to cell integrity
and cohesion of the organ lining [18]. Te loss of cohesion between
tight junctions could lead to dysplastic changes, which may eventually
transform into cancer [19].
It must be noted that a relationship between TJ proteins and
epithelial cancers is complex. An intact and functional TJ complex
acts as a barrier to the initiation and progression of epithelial cancers
by regulating important processes such as cell polarity, cell fate and
cell movement. However, any imbalance in the protein components
of this complex (whether increased or decreased) might disrupt the
homeostatic control required to maintain the tissue in its diferentiated
state. Te imbalance can also alter cell-cell and cell-extracellular
matrix interactions, and cause disordered organ lining that makes
cells chronically leaky to mitogens and growth factors. Together, these
events can promote cancer formation in premalignant epithelial tissues
[7]. Disruptive changes in TJ complex can also alter cell adhesion, free
tumor cells from both neighboring cells and the underlying matrix;
and confer onto them a migratory or invasive characteristics [20].
Te role of individual TJ proteins in this process is suggested by the
following few examples from a large body of evidence. Te role of
claudin-1 in the control of cell fate is indicated by increased expression
in senescent epithelial cells and reduced expression in invasive cancers
[21]. Decreased ZO-1 expression correlates with decreased glandular
diferentiation of breast tumor specimens [22]. ZO-1 and ZO-2 also
regulate cell cycle progression and proliferation in a cell density-
dependent manner through transcription factors such as ZONAB [23].
A large majority of cancers afecting elderly population are
epithelial, and display dysregulated cell-cell adhesion. With better
understanding of the factors and mechanisms involved in dysregulated
cell-cell adhesion, it is becoming apparent that therapies specifcally
directed at restoring normal TJ function might be benefcial in halting
the progression of epithelial tumors and in restoring normal cell-cell
adhesion patterns. Unfortunately, the delivery of the TJ-targeting
therapeutic agents to the site of action can pose a major problem.
Te agent must traverse epithelial and/or endothelial barriers to
reach the site of action. Since the TJ is the primary regulator of
paracellular transport across such cells, successful drug delivery may
require modulation of TJ proteins to allow drug molecules to pass
*Corresponding author: Girish V Shah, Department of Pharmacology, University
of Louisiana, Monroe, LA 71291, USA, E-Mail: shah@ulm.edu
Received August 17, 2012; Accepted August 20, 2012; Published August 23,
2012
Citation: Shah GV (2012) Restoration of Tight-Junction Function: A New
Therapeutic Approach for the Treatment of Cancer. Biochem Pharmacol 1:e130.
doi:10.4172/2167-0501.1000e130
Copyright: © 2012 Shah GV, et al. This is an open-access article distributed under
the terms of the Creative Commons Attribution License, which permits unrestricted
use, distribution, and reproduction in any medium, provided the original author and
source are credited.
Restoration of Tight-Junction Function: A New Therapeutic Approach for
the Treatment of Cancer
Girish V Shah*
Department of Pharmacology, University of Louisiana, Monroe, LA 71291, USA
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ISSN: 2167-0501
Biochemistry & Pharmacology: Open
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