Copyright © Italian Federation of Cardiology. Unauthorized reproduction of this article is prohibited.
Chemotherapy cardiotoxicity: cardioprotective drugs and
early identification of cardiac dysfunction
Daniela Di Lisi
a
, Giuseppe Leggio
a
, Giuseppe Vitale
a
, Salvatore Arrotti
a
,
Rosanna Iacona
a
, Riccardo Maria Inciardi
a
, Domenico Nobile
a
,
Francesca Bonura
a
, Giuseppina Novo
a
, Antonio Russo
b
and Salvatore Novo
a
Background Chemotherapy cardiotoxicity is an emerging
problem and it is very important to prevent cardiac
dysfunction caused by anticancer drugs. The aim of this
study was to assess the alterations of the cardiac function
induced by chemotherapy in a follow-up of 2 years and to
evaluate the cardioprotective role of angiotensin-converting
enzyme inhibitors (ACEIs) in the prevention of cardiac
dysfunction.
Methods A prospective study was carried out using
patients with breast cancer (85 women; median age
57 W 12 years) and other inclusion and exclusion criteria. On
the basis of treatment, patients were divided into six groups:
fluorouracil-epirubicincyclophosphamide, FEC (group A);
FEC and trastuzumab (B); trastuzumab (C); FEC and
taxotere (D); FEC, paclitaxel and trastuzumab (E); and
chemotherapy and cardioprotective drugs (F). Cardiological
evaluation including electrocardiogram and conventional
echocardiogram with tissue Doppler imaging (TDI) was
carried out at T0 (before starting chemotherapy), T1 (after
6 months from the start of chemotherapy) and T2 (2 years
after the end of chemotherapy).
Results Significant changes in the TDI parameters of
systolic and diastolic function were observed at T1 and T2 in
all patients. A significant reduction of left ventricular ejection
fraction (LVEF) was observed only at T2. In the patients
treated with ACEI (F), these changes were less significant
than in other groups and they do not have significant
changes in the indices of diastolic function.
Conclusion TDI is more sensitive than conventional
echocardiogram in the early diagnosis of cardiac
dysfunction and ACEIs seem to have an important role in the
prevention of cardiotoxicity.
J Cardiovasc Med 2014, 16:000–000
Keywords: angiotensin-converting enzyme inhibitor, cardiotoxicity,
chemotherapy, prevention, tissue Doppler imaging
a
Department of Biomedicine, Internal Medicine and Specialities (DIBIMIS),
Division of Cardiology and
b
Division of Oncology, University Hospital
‘P.Giaccone’, University of Palermo, Palermo, Italy
Correspondence to Giuseppe Leggio, MD, Department of Biomedicine, Internal
Medicine and Specialities (DIBIMIS), Division of Cardiology, University Hospital
‘P.Giaccone’, University of Palermo, Palermo 90127, Italy.
E-mail: giuseppeleggio1988@gmail.com
Received 30 January 2014 Revised 22 September 2014
Accepted 23 September 2014
Introduction
Chemotherapy cardiotoxicity is an emerging problem.
Some drugs, such as anthracyclines and other biological
agents, can cause cardiovascular complications (left ven-
tricular dysfunction, heart failure, myocardial ischemia,
hypertension, arrhytmias, pericarditis, cardiac tampo-
nade).
1
Anthacycline-induced cardiotoxicity has been
categorized into acute, early-onset chronic progressive
and late-onset chronic progressive.
2
Late anthracycline
cardiotoxicity is cumulative, dose related and high
dosages can result in congestive heart failure and left
ventricular dysfunction.
3
Usually, cardiac damage caused
by anthracycline is irreversible (Type I cardiotoxicity).
Trastuzumab induces predominantly reversible dysfunc-
tion (Type II cardiotoxicity).
4
This classification system
does have limitations; for example, trastuzumab, a Type
II drug, can trigger irreversible cardiac damage in patients
with severe preexisting cardiac disease or potentiate
anthracycline Type I cardiotoxicity. In Type I cardio-
toxicity, usually pathophysiology is related to cell loss,
and in Type II, cellular dysfunction (mitochondrial and
protein alterations) underlies the reversible damage.
5
Thus, it is very important that the early diagnosis of left
ventricular dysfunction induced by anticancer drugs
using tissue echocardiographic parameters [such as tissue
Doppler imaging (TDI) and speckle tracking] is more
sensitive than conventional echocardiography and the
prevention of severe forms of cardiac dysfunction using
early cardioprotective drugs [such as angiotensin-
converting enzyme inhibitor (ACEI), angiotensin recep-
tor blockers (ARBs) and beta-blockers] when subclinical
cardiotoxicity has been identified.
6
The aim of this study was to assess the alterations of the
cardiac function induced by chemotherapy in a follow-up
of 2 years (using conventional echocardiographic
parameters associated with tissue Doppler parameters)
and to evaluate the protective role of drugs (ACEI, ARBs
and beta-blockers) in the prevention of severe forms of
cardiac dysfunction.
Original article
1558-2027 ß 2014 Italian Federation of Cardiology DOI:10.2459/JCM.0000000000000232
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