Research Article
Doxycycline and Benznidazole Reduce the Profile of Th1,
Th2, and Th17 Chemokines and Chemokine Receptors in
Cardiac Tissue from Chronic Trypanosoma cruzi-Infected Dogs
Guilherme de Paula Costa,
1
Laís Roquete Lopes,
1
Maria Cláudia da Silva,
2
Aline Luciano Horta,
1
Washington Martins Pontes,
1
Cristiane M. Milanezi,
2
Paulo Marcos da Mata Guedes,
3
Wanderson Geraldo de Lima,
1,4
Richard Schulz,
5
João Santana da Silva,
2
and Andre Talvani
1,4,6
1
Programa de P´ os-Graduac ¸˜ ao em Ciˆ encias Biol´ ogicas/NUPEB, Universidade Federal de Ouro Preto, Ouro Preto, MG, Brazil
2
Faculdade de Medicina de Ribeir˜ ao Preto, USP, Ribeir˜ ao Preto, SP, Brazil
3
Universidade Federal do Rio Grande do Norte Federal, Natal, RN, Brazil
4
Departamento de Ciˆ encias Biol´ ogicas, Universidade Federal de Ouro Preto, Ouro Preto, MG, Brazil
5
Departments of Pediatrics & Pharmacology, Cardiovascular Research Centre, University of Alberta, Edmonton, AB, Canada
6
Programa de P´ os-Graduac ¸˜ ao em Sa´ ude e Nutric ¸˜ ao, Universidade Federal de Ouro Preto, Ouro Preto, MG, Brazil
Correspondence should be addressed to Andre Talvani; talvani@nupeb.ufop.br
Received 2 April 2016; Revised 14 July 2016; Accepted 4 August 2016
Academic Editor: Sandra Helena Penha Oliveira
Copyright © 2016 Guilherme de Paula Costa et al. Tis is an open access article distributed under the Creative Commons
Attribution License, which permits unrestricted use, distribution, and reproduction in any medium, provided the original work is
properly cited.
Chemokines (CKs) and chemokine receptors (CKR) promote leukocyte recruitment into cardiac tissue infected by the Trypanosoma
cruzi. Tis study investigated the long-term treatment with subantimicrobial doses of doxycycline (Dox) in association, or not, with
benznidazole (Bz) on the expression of CK and CKR in cardiac tissue. Tirty mongrel dogs were infected, or not, with the Berenice-
78 strain of T. cruzi and grouped according their treatments: (i) two months afer infection, Dox (50 mg/kg) 2x/day for 12 months;
(ii) nine months afer infection, Bz (3,5mg/Kg) 2x/day for 60 days; (iii) Dox + Bz; and (iv) vehicle. Afer 14 months of infection,
hearts were excised and processed for qPCR analysis of T1 (CCL2, CCL3, CCL4, CCL5, CXCL9, and CXCL11), T2 (CCL1, CCL17,
CCL24, and CCL26), T17 (CCL20) CKs, T1 (CCR5, CCR6, and CXCR3), and T2/T17 (CCR3, CCR4, and CCR8) CKR, as well
as IL-17. T. cruzi infection increases CCL1, CCL2, CCL4, CCL5, CCL17, CXCL10, and CCR5 expression in the heart. Dox, Bz, or Dox
+ Bz treatments cause a reversal of CK and CKR and reduce the expression of CCL20, IL-17, CCR6, and CXCR3. Our data reveal
an immune modulatory efect of Dox with Bz, during the chronic phase of infection suggesting a promising therapy for cardiac
protection.
1. Introduction
Chemokines are low molecular weight proteins that promote
leukocyte trafcking in homeostasis and infammatory pro-
cesses. Chronic infammation is usually characterized by the
persistence of leukocyte infltration into the infammatory
site driven by chemokine production [1–3]. In particular,
Trypanosoma cruzi infection is a well-known parasite disease
where the presence of this protozoan triggers activation and
continued leukocyte infltration into the muscle tissues in
order to eliminate it [4–6]. Since the stimulus persists over
months, years, or decades, cell infltration conducted by T1
and T2-like chemokines and their receptors may lead to loss
of tissue’s architecture and function, in some cases causing
severe disability, especially in the heart [7, 8].
Afer the interaction between T. cruzi and mammalian
host cells, the activation of innate resident macrophages/
neutrophils combined with the mobilization of natural killer
Hindawi Publishing Corporation
Mediators of Inflammation
Volume 2016, Article ID 3694714, 11 pages
http://dx.doi.org/10.1155/2016/3694714