O'Beirne et al. Journal of Experimental & Clinical Cancer Research 2010, 29:48
http://www.jeccr.com/content/29/1/48
Open Access RESEARCH
BioMed Central
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Research
Generation of functional CD8+ T Cells by human
dendritic cells expressing glypican-3 epitopes
James O'Beirne
1,3
, Farzin Farzaneh
2
and Phillip M Harrison*
1
Abstract
Background: Glypican 3 (GPC-3) is an oncofoetal protein that is expressed in most hepatocellular carcinomas (HCC).
Since it is a potential target for T cell immunotherapy, we investigated the generation of functional, GPC-3 specific T
cells from peripheral blood mononuclear cells (PBMC).
Methods: Dendritic cells (DC) were derived from adherent PBMC cultured at 37°C for 7 days in X-Vivo, 1% autologous
plasma, and 800 u/ml GM-CSF plus 500 u/ml IL-4. Immature DC were transfected with 20 μg of in vitro synthesised GPC-
3 mRNA by electroporation using the Easy-ject plus system (Equibio, UK) (300 V, 150 μF and 4 ms pulse time), or pulsed
with peptide, and subsequently matured with lipopolysaccharide (LPS). Six predicted GPC-3 peptide epitopes were
synthesized using standard f-moc technology and tested for their binding affinity to HLA-A2.1 molecules using the cell
line T2.
Results: DC transfected with GPC-3 mRNA but not control DC demonstrated strong intracellular staining for GPC-3 and
in vitro generated interferon-gamma expressing T cells from autologous PBMC harvested from normal subjects. One
peptide, GPC-3
522-530
FLAELAYDL, fulfilled our criteria as a naturally processed, HLA-A2-restricted cytotoxic T
lymphocyte (CTL) epitope: i) it showed high affinity binding to HLA-A2, in T2 cell binding assay; ii) it was generated by
the MHC class I processing pathway in DC transfected with GPC-3 mRNA, and iii) HLA-A2 positive DC loaded with the
peptide stimulated proliferation in autologous T cells and generated CTL that lysed HLA-A2 and GPC-3 positive target
cells.
Conclusions: These findings demonstrate that electroporation of GPC-3 mRNA is an efficient method to load human
monocyte-derived DC with antigen because in vitro they generated GPC-3-reactive T cells that were functional, as
shown by interferon-gamma production. Furthermore, this study identified a novel naturally processed, HLA-A2-
restricted CTL epitope, GPC-3
522-530
FLAELAYDL, which can be used to monitor HLA-A2-restricted CTL responses in
patients with HCC. Further studies are required to investigate whether anti-GPC-3 immunotherapy has a role in the
treatment of GPC-3 dependent tumours, such as HCC.
Background
Increasing evidence suggests that immune responses play
an important role in the control of cancer and manipula-
tion of the immune system to recognize and attack cancer
cells may be a valuable form of therapy [1]. Hepatocellu-
lar carcinoma (HCC), which is the third most common
cause of cancer death world-wide [2], is a potential target
for immunotherapy [3] because there are numerous doc-
umented cases of spontaneous regression [4] and the
presence of cytotoxic tumour infiltrating lymphocytes
(TIL) at histological examination is associated with a bet-
ter prognosis after liver resection or transplantation [5].
Infusion of T lymphocytes, activated with anti CD3 and
interleukin 2 (IL2), improved disease-free survival after
HCC resection, suggesting a role for T cell immunother-
apy in this setting [6]. However, current methods of isola-
tion and in vitro expansion of T lymphocytes are
cumbersome and expensive, and the durability of any
anti-tumour immune response induced by administra-
tion of non-antigen specific, in vitro expanded T cells is
unknown [7].
* Correspondence: phillip.harrison@kcl.ac.uk
1
Department of Liver Studies & Transplantation, Kings College London,
Denmark Hill Campus, Bessemer Road, London, SE5 9RS, UK
Full list of author information is available at the end of the article