cancers
Article
HGF/MET Axis Induces Tumor Secretion of Tenascin-C and
Promotes Stromal Rewiring in Pancreatic Cancer
Chiara Modica
1
, Martina Olivero
1,2
, Francesca Zuppini
1,2
, Melissa Milan
1
, Cristina Basilico
1,
*
and Elisa Vigna
1,2,
*
Citation: Modica, C.; Olivero, M.;
Zuppini, F.; Milan, M.; Basilico, C.;
Vigna, E. HGF/MET Axis Induces
Tumor Secretion of Tenascin-C and
Promotes Stromal Rewiring in
Pancreatic Cancer. Cancers 2021, 13,
3519. https://doi.org/10.3390/
cancers13143519
Academic Editor: Guido Eibl
Received: 30 April 2021
Accepted: 10 July 2021
Published: 14 July 2021
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1
Candiolo Cancer Institute, FPO-IRCCS, 10060 Candiolo, Italy; modicachiara89@gmail.com (C.M.);
martina.olivero@ircc.it (M.O.); francesca.zuppini@unito.it (F.Z.); melissa.milan@ircc.it (M.M.)
2
Department of Oncology, University of Turin, 10060 Candiolo, Italy
* Correspondence: cribasilico@gmail.com (C.B.); elisa.vigna@ircc.it (E.V.); Tel.: +39-011-993-3228 (C.B. & E.V.)
Simple Summary: It has been previously shown that activation of the MET receptor by its ligand,
the hepatocyte growth factor (HGF), modulates the tumor-stroma cross-talk in models of pancreatic
cancer. We now wish to cast light on the molecular mechanisms by which this ligand/receptor
pair sustains the interaction between cancer cells and the tumor microenviroment. To this end, we
compared data obtained by large-scale analysis of gene expression in pancreatic cancer cells grown
in the presence of HGF versus cells grown in the presence of HGF and treated with specific inhibitors
of HGF/MET signaling. By clustering differentially expressed genes according to functional groups,
we identified candidate genes involved in the process. Among these, tenascin C was selected due
to its activity in sustaining the malignant phenotype. Our results highlight a new role for tenascin
C, which could represent the operative arm through which MET promotes activation of the stromal
compartment in pancreatic cancer.
Abstract: Pancreatic ductal adenocarcinoma is an aggressive tumor characterized by the presence of
an abundant stromal compartment contributing significantly to the malignant phenotype. Pancreatic
stellate cells are peculiar fibroblasts present in the stroma and represent the predominant source of
extracellular matrix proteins, pro-inflammatory cytokines, and growth factors, including hepatocyte
growth factor (HGF). Exploiting a co-culture system of human pancreatic stellate cells and cancer
cells, we demonstrated that fibroblast activation was reduced upon HGF/MET axis inhibition.
To unveil the signaling pathways sustaining stroma modulation orchestrated by MET activation
in the tumor, we analyzed the gene expression profile in pancreatic cancer cells stimulated with
HGF and treated with HGF/MET inhibitors. Transcriptome analysis showed that, among all the
genes modulated by HGF, a subset of 125 genes was restored to the basal level following treatment
with the inhibitors. By examining these genes via ingenuity pathway analysis, tenascin C emerged
as a promising candidate linking MET signaling and tumor microenvironment. MET-dependent
tenascin C modulation in pancreatic cancer cells was validated at RNA and protein levels both
in vitro and in vivo. In conclusion, this work identifies tenascin C as a gene modulated by MET
activation, suggesting a role in MET-mediated tumor-stroma interplay occurring during pancreatic
tumor progression.
Keywords: pancreatic ductal adenocarcinoma; tumor microenvironment; hepatocyte growth factor;
MET oncogene; tenascin C; metastasis
1. Introduction
Pancreatic ductal adenocarcinoma (PDAC) is the most common type of pancreatic
cancer and is characterized by highly aggressive behavior [1]. According to the PDAC
progression model, invasive adenocarcinoma arises from a well-defined duct lesion, called
a pancreatic intraepithelial neoplasia, which evolves into a malignant adenocarcinoma
Cancers 2021, 13, 3519. https://doi.org/10.3390/cancers13143519 https://www.mdpi.com/journal/cancers