Area Under Curve Method Development for Etodolac in Bulk and Tablet dosage
form
Vaibhav G Bhamare
1*
, Renuka R Joshi
2
, RD Amrutkar
3
1
Department of Research Scholar, Bhupal Nobles University, Udaipur, India;
2
Department of Pharmaceutical Quality Assurance,
Mahatma Gandhi Vidyamandir’s Pharmacy College, Panchavati, Nashik, India;
3
Department of Pharmaceutical Chemistry, MGV’s
SPH College of Pharmacy, Malegaon, India
ABSTRACT
A simple,precise, rapid and economical spectroscopic method has been developed for the determination of Etodolac
in bulk and tablet dosage form. In methanol Etodolac shows absorbance maxima at 281nm. Method used was area
under curve in which area incorporated in the wavelength range of 275nm-285nm.Etodolac obeys Beer’s law in
concentration range 0-60µg/ml. Calibration curves were plotted at selected wavelengths and it was found to be linear
(r2=0.9997) Linearity for detector response was observed in the concentration range of 5-30µg/ml. The recovery
studies established accuracy of the proposed method and results validated according to ICH guideline. Precision and
Accuracy studies were carried out and results were satisfactory. Robustness of the given method was studied by using
two wavelength, 279nm and 283nm respectively. Results were found satisfactory and reproducible. The developed
method was successfully applied to estimate the amount of Etodolac in pharmaceutical formulation.
Keywords: Area under curve; accuracy, precision; spectroscopic method.
INTRODUCTION
Etodolac is non steroidalanti inflammatory drug which is
belongs to pyranocarboxylic acid class developed in the 1970s. It
blocks production of certain natural substances that causes
inflammation [1]. Etodolac is chemically 1, 8-Diethyl-1, 3, 4, 9-
tetrahydropyrone (3, 4-b) indole -1-acetic acid. Molecular formula
of Etodolac is C17H21No3 [2].Cox present in two separate
entities, one is Cox-1 and other is Cox-2[3, 4]. It inhibits
synthesis of peripheral prostaglandins, by decreasing the activity
of the Cox enzyme. Cox-1 protect the integrity of the stomach
lining and sustain normal renal function in a kidney .Cox-2
plays a vital role in both control of cell growth and inflammation
[5].Peak serum concentration achieved within 2 hours of oral
administration of Etodolac 200mg and 400mg respectively [6] It
is rapidly metabolized in the liver, followed by renal elimination
as the primary route of excretion [7].
It is used for rheumatoid arthritis and osteoarthritis,
postoperative pain and inflammation [8].It is used as anti-
inflammatory agent, analgesic antipyretic and cyclooxygenase
inhibitor. Etodolac is official in the United States
Pharmacopoeia and British Pharmacopoeia [9].
Method development is the process of verifying that an analytical
method is good enough for exercise to measure the
concentration of an API in a particular compounded dosage
form which allow basicmeasures to be employed to confirm that
an analysis procedure, precisely and consistently will deliver a
trustworthy measurement of an active ingredient in a
compounded preparation [10].Primary purpose of method
development to generate date regarding efficiency, safety,
impurity, stability (that shows degradation of product),
bioavailability and the effect of manufacturing parameter (that
shows steadiness of the product) [11].
MATERIALS AND METHODS
The spectrophotometric analysis was carried out using a
Labindia UV-3000 Uv/Vis spectrophotometer with 1 cm
matched quartz cell. The spectra were obtained with the
instrumental parameters as follows:Wavelength range (nm):
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ISSN: 2329-6631
Journal of Developing Drugs
Research Article
*Corresponding author: Vaibhav G Bhamare, Department of Research Scholar, Bhupal Nobles University, Udaipur, India, Tel: 7588176846; E-mail:
vaibhav.bhamre@gmail.com
Received date: April 02, 2021; Accepted date:April 16, 2021; Published date: April 23, 2021
Citation: Bhamarre VG, Joshi RR, Amrutkar RD (2021) AreaUnder Curve Method Development for Etodolac in Bulk and Tablet dosage form. J
Develop Drugs. 10:207.
Copyright: ©2021 Bhamare VG, et al. This is an open-access article distributed under the terms of the Creative Commons Attribution License,
which permits unrestricted use, distribution, and reproduction in any medium, provided the original author and source are credited.
J Develop Drugs, Vol.10 Iss.3 No:1000207 1