www.thelancet.com/neurology Vol 18 June 2019 539
Articles
Lancet Neurol 2019; 18: 539–48
See Comment page 515
Department of Cerebrovascular
Medicine, National Cerebral and
Cardiovascular Centre, Osaka,
Japan (K Toyoda MD,
T Yamaguchi MD); Clinical
Research Centre for Medicine,
International University of
Health and Welfare, Tokyo,
Japan (S Uchiyama MD); Centre
for Brain and Cerebral Vessels,
Sanno Hospital and Sanno
Medical Centre, Tokyo, Japan
(S Uchiyama); Department of
Neurology, University of
California, San Francisco, CA,
USA (J D Easton MD);
Department of Neurological
Science, Graduate School of
Medicine, Nippon Medical
School, Tokyo, Japan
(K Kimura MD); Department of
Neurology, Tokyo Saiseikai
Central Hospital, Tokyo, Japan
(H Hoshino MD); Department of
Neurosurgery, Kobe City
Medical Centre General
Hospital, Kobe, Japan
(N Sakai MD); Clinical Research
Institute and Department of
Cerebrovascular Medicine and
Neurology, National Hospital
Organisation Kyushu Medical
Centre, Fukuoka, Japan
(Y Okada MD); Department of
Neurology (K Tanaka MD) and
Division of Biostatistics and
Clinical Epidemiology
(H Origasa PhD), University of
Toyama, Toyama, Japan;
Department of Neurology, Senri
Chuo Hospital, Toyonaka, Japan
(H Naritomi MD); Department of
Neurosurgery, Hokkaido
University Graduate School of
Medicine, Sapporo, Japan
(K Houkin MD); Department of
Neurology, Ichinomiya Nishi
Hospital, Ichinomiya, Japan
(K Yamaguchi MD); Department
of Neurosurgery, Kushiro Rosai
Hospital, Kushiro, Japan
(M Isobe MD); and Headquarters
of the Iseikai Medical
Corporation, Osaka, Japan
(K Minematsu MD)
Dual antiplatelet therapy using cilostazol for secondary
prevention in patients with high-risk ischaemic stroke in
Japan: a multicentre, open-label, randomised controlled trial
Kazunori Toyoda, Shinichiro Uchiyama, Takenori Yamaguchi, J Donald Easton, Kazumi Kimura, Haruhiko Hoshino, Nobuyuki Sakai,
Yasushi Okada, Kortaro Tanaka, Hideki Origasa, Hiroaki Naritomi, Kiyohiro Houkin, Keiji Yamaguchi, Masanori Isobe, Kazuo Minematsu, on behalf
of the CSPS.com Trial Investigators
Summary
Background Although dual antiplatelet therapy with aspirin and clopidogrel reduces early recurrence of ischaemic
stroke, with long-term use this type of therapy is no longer efective and the risk of bleeding increases. Given that
cilostazol prevents stroke recurrence without increasing the incidence of serious bleeding compared with aspirin, we
aimed to establish whether dual antiplatelet therapy involving cilostazol is safe and appropriate for long-term use.
Methods In a multicentre, open-label, randomised controlled trial across 292 hospitals in Japan, patients with high-
risk non-cardioembolic ischaemic stroke identifed on MRI were randomly assigned to two groups in a 1:1 ratio to
receive monotherapy with either oral aspirin (81 or 100 mg, once per day) or clopidogrel (50 or 75 mg, once per day)
alone, or a combination of cilostazol (100 mg, twice per day) with aspirin or clopidogrel. Randomisation was done
centrally (using block randomisation with a block size of six per each participating hospital) through a web-based
registration system and was done by EPS Corporation. The patients were required to have at least 50% stenosis of a
major intracranial or extracranial artery or two or more of the vascular risk factors. Trial medication was continued for
half a year or longer, for a maximum of 3·5 years. The primary efcacy outcome was the rate of frst recurrence of
symptomatic ischaemic stroke. Safety outcomes were severe or life-threatening bleeding; any adverse events; serious
adverse events; and any bleeding events. Efcacy analyses were done in the intention-to-treat population and safety
analyses were done in the as-treated population. This trial was registered with ClinicalTrials.gov (number
NCT01995370) and UMIN Clinical Trials Registry (number 000012180).
Findings Participants were recruited from Dec 13, 2013, to March 31, 2017. 932 patients assigned to the dual therapy
group and 947 patients assigned to the monotherapy group were included in the intention-to-treat analysis. The trial
was stopped after the enrolment of 1884 patients of an anticipated 4000 patients because of the delay in recruitment.
Ischaemic stroke recurred in 29 (3%) of 932 patients (annualised rate 2·2%) on dual therapy including cilostazol and
64 (7%) of 947 patients (annualised rate 4·5%) on monotherapy during a median 1·4 years follow-up (hazard ratio
[HR] 0·49, 95% CI 0·31–0·76, p=0·0010). Severe or life-threatening bleeding occurred in eight patients (annualised
rate 0·6%) on dual therapy and 13 patients (annualised rate 0·9%) on monotherapy (HR 0·66, 95% CI 0·27–1·60,
p=0·35). Occurrence of any type of adverse event was similar between the groups (255 [28%] of 910 patients in the
dual therapy group vs 219 [24%] of 921 patients in the monotherapy group); as was occurrence of serious adverse
events (87 [10%] vs 142 [15%]) and bleeding events (38 [4%] vs 33 [4%]). Gastrointestinal bleeding, which afected
nine (<1%) of 910 patients in the monotherapy group and nine (<1%) of 921 patients in the dual therapy group, was
the most common type of bleeding.
Interpretation The combination of cilostazol with aspirin or clopidogrel had a reduced incidence of ischaemic stroke
recurrence and a similar risk of severe or life-threatening bleeding compared with treatment with aspirin or
clopidogrel alone in patients at high risk for recurrent ischaemic stroke.
Funding Otsuka Pharmaceutical.
Copyright © 2019 Elsevier Ltd. All rights reserved.
Introduction
Patients with non-cardioembolic ischaemic stroke have a
higher risk of recurrence when they have carotid steno-
sis,
1
intracranial arterial stenosis,
2
or multiple vascular
risk factors than when they do not have these com-
plications.
3,4
For such patients, comprehensive preventive
therapy, including antiplatelet medication, has been
proven benefcial. However, newer antiplatelet agents
that are promising for patients with coronary artery
disease and have been in commercial use for around
10 years, such as ticagrelor and prasugrel, did not show
advantages over conventional antiplatelet agents for
patients with stroke in randomised controlled trials
(RCTs).
5,6