Sustainable Chemistry and Pharmacy 18 (2020) 100325
Available online 11 September 2020
2352-5541/© 2020 Elsevier B.V. All rights reserved.
Fabrication and evaluation of pH-sensitive biocompatible microwave
irradiated moringa barkgum-carrageenan (MOG-CRG-IPN) interpenetrating
isotropic polymeric network for controlled delivery of pharmaceuticals
Debjani Roy , Trishna Bal
*
, Sabyasachi Swain
Department of Pharmaceutical Sciences and Technology, Birla Institute of Technology, Mesra, Ranchi, 835215, India
A R T I C L E INFO
Keywords:
Moringa bark gum (MOG)
Carageenan(CRG)
Microwave irradiation
Controlled release
ABSTRACT
In the present research, pH-sensitive interpenetrating polymeric network are prepared by interpenetration of two
natural polysaccharides Moringa bark gum(MOG) and Carrageenan (CRG) by use of microwave irradiation as
interpenetrating polymeric network (IPN) and characterized using fourier transform infrared spectroscopy
(FTIR), x-ray diffraction (XRD), thermogravimetric studies (TGA) and 13C nuclear magnetic resonance (13C
NMR) and the surface topography, indepth pore size as well as the interior architecture of the material were
confrmed by scanning electron microscopy(SEM) and atomic force microscopy (AFM).The contact angle mea-
surement by optical contact angle (OCA) indicated that the increase in MOG content increased the water
retention capacity thereby maintaining the structural integrity of the polymeric network. The pH sensitivity at
pH 2,7.4 & 9.2 and swelling studies helped in optimizing the best grade F7.The swelling kinetics of F7 followed
second order kinetics. The biodegradability studies were done using soil burial method.The drug release from F7
was found to 88.17% for 8 h interval. The material proved to be hemocompatible. These studies indicated that
MOG-CRG-IPN (F7) can be effectively used as an effcient controlled delivery device and can be explored as
biomaterial.
1. Introduction
Stimuli sensitive interpenetrating polymeric network systems(IPNs)
are gaining importance as effcient drug delivery device (Wells and
Harris, 2019) as well as polymeric scaffolds. An interpenetrating poly-
mer network is a system of more than one polymer where at least one
polymer is crosslinked in the immediate presence of other polymer
(Zhao, 2012), thereby retaining the individual characteristics of the
polymers used in the process.Various natural polymers along with
combinations of synthetic polymers are used for the preparation of IPN
(Wells and Harris, 2019; Swain and Bal, 2019a). Moringa Bark Gum
(MOG) obtained from the bark of Moringa oleifera is a reddish brown
polysaccharide having very good swelling properties due to presence of
numerous hydroxyl groups on the polymer backbone and consists of
arabinose, galactose and glucoronic acid in the ratio of 10:7:2 (Panda
et al., 2006), whereas Carrageenan (CRG), obtained from red sea weed is
an important natural polysaccharide due to its thickening, emulsifying
as well as thermo-reversible gelling properties having higher molecular
weight with a curly-helical structure in which 3,6-anhydrogalactose and
are attached with D-galactose by α-1,3 and β-1,4 glycoside linkage and
through crosslinking a double helix structure can be formed due to the
presence of sulfate group in the spiral chains of CRG (Swain and Bal,
2019a).The blend of CRG with MOG aided by microwave irradiation
facilitates the crosslinks between MOG and CRG by virtue of hydrogen
bond formation between sulfate groups of CRG and the hydroxyl groups
of MOG thus forming a double helical structure by helic entanglement.
Due to this formation of double helix within the crosslinked polymer
blend, the swelling property of the MOG-CRG-IPN system is also
enhanced which is an most important property for drug loading (Swain
and Bal, 2019a). In the feld of tissue engineering also, such IPN plays a
signifcant role as scaffold which is already studied earlier (Swain and
Bal, 2019b), for wound repair (Dhandayuthapani and YoshidaTor-
uMaekawa, 2011), burn, accidents or severe trauma, where the tissue
grows on the polymeric backbone leaving the site of injury without any
scars.These materials as scaffolds can mimic the extracellular matrix,
thereby provoking the cells to adapt to proliferation and differentiaton
(Malafaya et al., 2007). The combination of CRG and MOG is unexplored
and no where in literature this combination has been applied for drug
* Corresponding author.
E-mail address: trishna.bal@gmail.com (T. Bal).
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Sustainable Chemistry and Pharmacy
journal homepage: http://www.elsevier.com/locate/scp
https://doi.org/10.1016/j.scp.2020.100325
Received 1 June 2020; Received in revised form 29 August 2020; Accepted 29 August 2020