Shukla et al Journal of Drug Delivery & Therapeutics. 2022; 12(4-S):264-269
ISSN: 2250-1177 [264] CODEN (USA): JDDTAO
Available online on 25.08.2022 at http://jddtonline.info
Journal of Drug Delivery and Therapeutics
Open Access to Pharmaceutical and Medical Research
Copyright © 2011-2022 The Author(s): This is an open-access article distributed under the terms of the CC BY-NC 4.0
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Open Access Full Text Article Review Article
Floating Microsponge: An Emerging Drug Delivery System
Mukesh Kumar Shukla
1
, Abadhesh Kumar Niranjan*
2
1
Research Scholar, Department of Pharmaceutics, Hygia Institute of Pharmaceutical Education and Research, Lucknow (U.P.) 226020, India
2
Associate Professor, Department of Pharmaceutics, Hygia Institute of Pharmaceutical Education and Research, Lucknow (U.P.) 226020, India
Article Info:
_____________________________________________
Article History:
Received 22 June 2022
Reviewed 13 August 2022
Accepted 21 August 2022
Published 25 August 2022
_____________________________________________
Cite this article as:
Shukla MK, Niranjan AK, Floating Microsponge:
An Emerging Drug Delivery System, Journal of
Drug Delivery and Therapeutics. 2022; 12(4-
S):264-269
DOI: http://dx.doi.org/10.22270/jddt.v12i4-s.5553
_____________________________________________
*Address for Correspondence:
Abadhesh Kumar Niranjan, Associate Professor,
Department of Pharmaceutics, Hygia Institute of
Pharmaceutical Education and Research, Lucknow
(U.P.) 226020, India
Abstract
___________________________________________________________________________________________________________________
Floating microsponges are a method to extend gastric residence time, there with the aid of using concentrated on
site-responsive medicament liberate withinside the top GIT for locally or systemic effect. Gastro retentive dosage
forms (GRDFs) are getting utilized from a totally long term to enhance treatment with numerous main medications.
Floating microsponge significantly enhances the therapy of stomach with the aid of using liberating the medication
locally and for that reason used for medication selecting at specific organ. This may be sustained over an extended
period of time. Floating drug delivery allow extended and non-stop release of the drug to the top a part of Gastro
intestinal tract and this expressively amplify the period of drug release and enhance pharmacokinetic of medication
which have slim healing window, with the aid of using this method dosing frequency and affected person compliance
is increased. A microsponge’s drug delivery system is a particularly cross-linkage, spongy, polymeric microsphere,
polymeric device consisting permeable microspheres. Microsponges are prepared with the aid of using numerous
techniques consisting of liquid-liquid suspension polymerization and quasi emulsion solvent diffusion method.
Microsponge,s preparations are strong over variety of pH 1 to 11; microsponge,s preparations are strong on the
temperature as much as 130
0
C well suited with maximum vehicles and ingredients. The present assessment
introduces microsponge,s technology at the side of its techniques of preparation, characterization, advantages,
evaluation and release mechanism of microsponge,s drug delivery system, advertised product and up to date studies
regarding microsponge.
Keywords: Floating microsponge, Oral administration, Controlled release, Quasi emulsion, Target release.
Contact No. 8317008539 E-mail: niranjanpharma88@gmail.com
1. Introduction:
1.1 Floating Drug Delivery System [FDDS]:
1,2,3
Oral route is maximum ideally path of drug delivery to easy
administration, pliability in preparation, low price and affected
person compliance. Oral controlled release drug delivery system
suggests a few restrictions associated with gastric emptying
time. Too rapid and variable gastric emptying should results in
insufficient drug release from dosage form into absorption
window main to low effectiveness of administered dose.
Floating drug delivery system become to put together the
presently awareness at the principle procedure of ability to float
to acquire gastric retention time. The modern tendencies of
FDDS together with the biological and approach variables
influencing gastric retention, strategies to format floating
structure, and their class and approach elements are enclosed in
detail. Gastroretentive system can remain within the gastric
region for several hours and as a result appreciably extend
gastric residence time of drug. Prolong gastric retention
enhances pliability of drugs which might be much less soluble in
an immoderate pH environment}, decreases drug wastages and
enhance bioavailability. FDDS has the main utility for the
delivery of local drugs to the stomach.
1.2 Basic Gastrointestinal tract Physiology:
4
For the improvement of Gastro-retentive drug delivery method
should have expertise of body structure of gastrointestinal tract.
Anatomically the stomach is split into 3 parts- (1) fundus, (2)
body and (3) antrum(pylorus) The contiguous element
fabricated from fundus and undigested material store in frame
so frame acts as reservoir, and antrum (pylorus) is the
responsible web page for mixing motion and acts as a pump,
cause gastric emptying.
Stomach Physiology:
2,4
The maximum crucial function of stomach is to process and to
convey the food. It act as a short‐time period storage reservoir,
enzymatic digestion started out in stomach wherein various
juices mix with food which is probably produced via gastric
smooth muscles and ensuing in liquefaction of food and it's
miles released for small intestine for in addition process].
Stomach is part of digestive system that's located amongst
oesophagus and small bowel. Structurally the wall of stomach is
alike to the alternative components of the digestive tube but
stomach has a likewise oblique layer of smooth muscle inside
the spherical layer which permits the motion inside the
stomach. When stomach is empty, it's far gotten smaller and its
mucous membrane and sub mucous membranes are thrown up
into wonderful folds known as rugae.