Rachmaniah et al. / Malaysian Journal of Fundamental and Applied Sciences Vol. 16, No. 5 (2020) 514-518
514
Orchidea Rachmaniah
*
, Galang Ramdhani Fitra Gama, Zandhika Alfi Pratama, Muhammad
Rachimoellah
Department of Chemical Engineering, Faculty of Industrial Technology, Institut Teknologi Sepuluh Nopember, 60111 Sukolilo, Surabaya, Indonesia
* Corresponding author: orchidea@its.ac.id
Article history
Received 8 April 2019
Revised 21 February 2020
Accepted 30 April 2020
Published Online 15 October 2020
Graphical abstract
Abstract
An antimicrobial photodynamic therapy (aPDT) is a local antimicrobial treatment which utilizes
a photosensitizer dye, visible light, and oxygen. It is considered as an alternative treatment for
bacterial or fungal resistance. In this treatmetn, a pure, stable and non-toxic natural
photosensitizer compound as a host cell which soluble in water and capable of producing
reactive photoproducts is required. Curcumin as a natural yellow-orange photosensitizer dye
with anti-inflammatory, anti-carcinogenic, anti-bacterial, and anti-infection activities is believed
to be safe for human consumption. Combining curcuminoids as a photosensitizer dye with
NADES as solvent instead of solving the low solubility drawback of curcuminoids in water, as
well as becoming a potential candidate of aPDT. However, an antimicrobial effect of dissolved
curcuminoids in NADES need to be studied first. Antimicrobial tests of curcuminoids to both of
Escherichia coli and Staphylococcus aureus using minimum inhibitory concentration (MIC) and
minimum bactericidal concentration (MBC) methods were conducted. Three NADES i.e. malic
acid-sucrose-water (MAS-H2O = 1:1:18); fructose-glucose-water (FG-H2O = 1:1:1); and
fructose-sucrose-water (FS-H2O = 2:1:15) were tested by applying nine different
concentrations of curcuminoids (2.00-4.00 mM). A blank of sample (no dissolved
curcuminoids) as well as a pure solution of each constituent compounds of NADES such
sucrose, malic acid, fructose, and glucose were also applied. Bacterial suspension approx. 10
8
cells/mL of 1 mL (24 h incubated at 37
o
C) was used for the test. MAS-H2O (1:1:18) shown the
most effective antimicrobial activity compared to both of FG-H2O (1:1:1) and FS-H2O (2:1:15).
The toxicity of MAS-H2O (1:1:18) to both E. coli and S. aureus may due to the low pH condition
of NADES itself since malic acid has high acidity (pH <3). Meanwhile, both other NADES
contains sugars, i.e. fructose, glucose, and sucrose, showing lower pH value (pH >5). Both on
the concentration of the curcuminoids and bacteria effects the observed toxicity.
Keywords: Antibacterial, curcuma, deep eutectic solvent, ionic liquid
© 2020 Penerbit UTM Press. All rights reserved
INTRODUCTION
Staphylococcus aureus strain has shown high resistance against
each new class of licensed antibiotics. It is recently reported that a strain
of S. aureus is resistant to vancomycin, a glycopeptide antibiotic
considered as a last line generation of antibiotics. The problem is made
more severe by social factors such as an inappropriate prescription of
antibiotics, or an excessive prescription of antibiotics leading to either
bacterial or fungal resistance. Moreover, more and more frequent
transmissions of microorganisms occur due to global traveling,
expansion of poverty among the population of the third world countries,
and by the large variety of mechanisms adopted by microbial cells, thus
increasing the resistance of the bacteria to external insults. This results
in a thickening of their outer wall, encoding of new proteins which
prevent the penetration of drugs, onset of mutants deficient in those
porin channels allowing the influx of externally added chemicals,
among others (Heger et al., 2014). Therefore, a comprehensive strategy
is required to resolve this problem, such as an alternative solution to
inactivate pathogens or bacteria.
A photochemical reaction among a photosensitizer (PS) or a dye,
visible light, and oxygen produces reactive oxygen species (ROS)
which is applied in antimicrobial photodynamic therapy (aPDT). The
produced ROS, free radicals and/or other reactive photoproducts may
cause damage to bacterial cell structures, which ultimately results in
bacterial inactivation. An alternative way to combat bacteria resistances
(Kumavat et al., 2013) is by overcoming the antibiotic resistances. A
visible light at an appropriate wavelength is used to excite the PS
molecule to produce superoxide radicals (type 1 reaction) or generate
singlet oxygen (type 2 reaction) (Kumavat et al., 2013) which
subsequently lead to the destruction of the bacterial cells by an
oxidative burst (Cieplik et al., 2018) of biomolecules such proteins,
lipids, and nucleic acids (Hamblin, 2016). It has been reported the
effectiveness of aPDT against Gram-positive, such Staphylococcus
aureus and Bacillus subtilis, and Gram-negative bacteria, such
RESEARCH ARTICLE
Antimicrobial effect of dissolved curcuminoid in natural deep
eutectic solvents (NADES) to Escherichia coli and Staphylococcus
aureus: A promising candidate for antimicrobial photodynamic
therapy (aPDT)