Vol.:(0123456789) 1 3
International Journal of Clinical Oncology
https://doi.org/10.1007/s10147-020-01771-1
ORIGINAL ARTICLE
YAP promotes self‑renewal of gastric cancer cells by inhibiting
expression of L‑PTGDS and PTGDR2
Qingli Bie
1,2
· Xiaozhe Li
1
· Shiqi Liu
3
· Xiao Yang
1
· Zhenwen Qian
1
· Rou Zhao
1
· Xiaobei Zhang
4
· Bin Zhang
1,2
Received: 8 May 2020 / Accepted: 10 August 2020
© Japan Society of Clinical Oncology 2020
Abstract
Introduction Cancer stem cells have been implicated angiogenesis of tumor and invasiveness, drug resistance in tumors.
Yes-associated protein 1 (YAP) owns carcinogenic roles in various organs, but the role of YAP in cancer stem cells of gas-
tric cancer (GC) remains unclear. In this study, we explored the function and mechanism of YAP in GC cancer stem cells.
Materials and methods, and results First, we confrmed that the expression of YAP mRNA and protein in GC tissues was
higher than in adjacent tissues by RT-PCR, western blot and immunohistochemistry. Immunofuorescence staining of the
GC tissues revealed that the region of YAP expression coincided with the region of expression of the cancer stem cell marker
SALL4 but did not overlap with that of the epithelial marker cytokeratin 14 (CK14). Additional research revealed that spheri-
cal cells expressed relatively high levels of YAP protein, and YAP overexpression reinforced self-renewal and expression of
stem cell markers in the GC cells. Knockdown the expression of YAP reversed this phenomenon. Second, we examined the
expression patterns of lipocalin-type prostaglandin D2 synthase (L-PTGDS) and prostaglandin D2 receptor 2 (PTGDR2) in
GC tissues and proved that there was negatively correlation between the expression of L-PTGDS and PTGDR2 and YAP in
GC tissues. Finally, we confrmed that YAP inhibited the expression of L-PTGDS and PTGDR2 by gain- and loss-of-function
experiments. Moreover, the overexpression of L-PTGDS and PTGDR2 suppressed the proliferation and self-renewal induced
by YAP in vitro and reversed the pro-tumor efect of YAP in vivo.
Conclusion Our results revealed a novel function of YAP and the mechanism underlying cancer stem cell regulation by YAP.
Keywords Yes-associated protein 1 · Prostaglandin D2 synthase · Prostaglandin D2 receptor 2 · Gastric · Cancer stem cell
Introduction
According to GLOBOCAN 2018, gastric cancer is the ffth
malignant tumor and the cause of the third tumor-related
death [1]. Gastric antrum cancers and gastric carcinomas are
most common cancer among GCs; however, the incidence of
gastroesophageal junction carcinomas is gradually increas-
ing [2, 3]. East Asian countries are considered areas with
high incidence of GCs, particularly Japan and China [4].
Despite the therapy of GCs has advanced in recent decades,
the prognosis of GC remains poor, because most patients
have reached the advanced stage when they are diagnosed
with gastric cancer, and current chemotherapy only improve
the survival time of patients [5]. Therefore, it is necessary
to identify novel targets and signaling molecules involved in
the tumorigenesis and progression of gastric cancer.
Yes-associated protein 1 (YAP) and transcriptional
coactivator with PDZ-binding motif (TAZ) are important
downstream transcription factors of the Hippo pathway [6].
Electronic supplementary material The online version of this
article (https://doi.org/10.1007/s10147-020-01771-1) contains
supplementary material, which is available to authorized users.
* Bin Zhang
zhb861109@163.com
1
Department of Laboratory Medicine, Afliated
Hospital of Jining Medical University, Jining Medical
University, 89 Guhuai Road, Jining 272000, Shandong,
People’s Republic of China
2
Institute of Forensic Medicine and Laboratory
Medicine, Jining Medical University, Jining, Shandong,
People’s Republic of China
3
Department of General Surgery, Afliated Hospital
of Jining Medical University, Jining, Shandong,
People’s Republic of China
4
Department of Central Laboratory, Afliated Hospital
of Jining Medical University, Jining, Shandong,
People’s Republic of China