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Original Research
Ergogenic Effects of 8 Days of Sceletium Tortuosum
Supplementation on Mood, Visual Tracking, and
Reaction in Recreationally Trained Men and Women
Jay R. Hoffman,
1
Irit Markus,
2
Gal Dubnov-Raz,
3
and Yftach Gepner
2
1
Department of Molecular Biology, Ariel University, Ariel, Israel;
2
Department of Epidemiology and Preventive Medicine, School of Public
Health, Sackler Faculty of Medicine and Sylvan Adams Sports Institute, Tel Aviv University, Tel Aviv, Israel; and
3
The Edmond and Lily
Safra Children’s Hospital, Sheba Medical Center, and Sackler Faculty of Medicine, Tel Aviv University, Tel Aviv, Israel
Abstract
Hoffman, JR, Marcus, I, Dubnov-Raz, G, and Gepner, Y. Ergogenic effects of 8 days of Sceletium tortuosum supplementation on
mood, visual tracking, and reaction in recreationally trained men and women. J Strength Cond Res 34(9): 2476–2481, 2020—
Sceletium tortuosum (ST) is a South African plant that has been reported to promote a sense of well-being in healthy individuals and
used in treating people with anxiety, stress, or depression. These studies have been conducted in middle-aged and older adults, but
no investigations have been performed in a healthy, young adult population. Thus, the purpose of this study was to examine the
effect of 8 days of ST extract (25-mg) supplementation on changes in reactive agility, visual tracking, and mood. Sixty recreationally
trained men (n 5 48) and women (n 5 12), between 20 and 35 years, were randomly assigned to 1 of 2 groups: ST or placebo (PL).
Subjects were tested on 2 occasions: before supplementation and 2-hours after supplementation on day 8. Subjects completed
a subjective questionnaire to assess alertness and energy using a visual analog scale (VAS). In addition, subjects completed the
Profile of Mood States questionnaire and performed reactive agility and visual tracking assessments. Significant improvements
were noted for ST in complex reactive performance that required subjects to respond to repeated visual stimuli with a cognitive load
compared with PL. However, no significant changes were noted between the groups in either VAS or total mood score. In addition,
no differences were observed in simple reaction assessments. The results of this study demonstrate an ergogenic benefit in
complex reactive tasks that include a cognitive load. However, in this subject population studied, no benefits in mood were
observed.
Key Words: dietary intervention, cognitive enhancer, reactive agility, performance, nutrition
Introduction
Sceletium tortuosum (ST) is a South African plant that has been
reported to promote a sense of well-being in healthy individuals
and used in treating people with anxiety, stress, or depression (7).
The physiological mechanism linked to its potential benefits
seems to be related to its role as a potent blocker of the serotonin
(5-HT) transporter and specifically act as an inhibitor of
phosphodiesterase-4 (PDE4) (10). Serotonin reuptake inhibitors
are generally used to treat depression, and recent evidence sug-
gests that PDE4 inhibitors can also be used as a potential treat-
ment option for depression (8). PDE4 inhibitors have also been
reported to attenuate proinflammatory cytokines (8). The po-
tential therapeutic benefit in the use of ST is that it may inhibit
both 5-HT and PDE4, potentially requiring a lower dose to
achieve desired efficacy, reducing the incidents of adverse events.
Serotonin is a neurotransmitter found in the brain that has an
important role in neuroplasticity (13). Dysfunction in neuro-
plasticity can result in learning and memory deficits, and it can
contribute to the pathophysiology of depression (13). Decreases
in serotonin as a result of an attenuated synthesis is thought to be
a cause of depression (16). Blocking the reuptake of 5-HT, thus
maintaining 5-HT concentrations, has been used as therapeutic
treatment for depression (17).
Phosphodiesterases (PDE) are a group of enzymes that catalyze
the hydrolysis of cyclic adenosine monophosphate (cAMP) (15).
Of the 11 PDEs, PDE4 has received much focus in neuro-
dysfunction because of its strong expression in the brain (9). The
immediate downstream effector of cAMP is protein kinase A
(PKA), which is activated upon cAMP binding and translocates to
the nucleus where it phosphorylates cAMP response element
binding protein (CREB). cAMP response element binding protein
is a transcription factor that binds to cAMP response element
promoter sites (2) located on specific CREB-mediated genes such
as brain-derived neurotrophic factor (BDNF), which can alter
synaptic function (6). Altered PDE4 signaling directly results in
cAMP alterations (9). The use of PDE4 inhibition as a therapeutic
option is to maintain the cAMP intracellular cascade. Others have
reported that PDE4 inhibition can also attenuate inflammatory
cytokines (12).
Terburg et al. (21) reported that a single administration of ST
extract (25 mg) can reduce anxiety-related amygdala reactivity
and attenuate amygdala-hypothalamus coupling, providing the
initial evidence that this plant is a dual PDE4 and 5-HT reuptake
inhibitor for the treatment of anxiety disorders and depression. A
subsequent investigation examined a 25-mg dose consumed for 3
weeks in middle-aged healthy men and women (4). Results from
this investigation demonstrated improvements in mood and in
Address correspondence to Dr. Jay R. Hoffman, jayho@ariel.ac.il.
Journal of Strength and Conditioning Research 34(9)/2476–2481
ª 2020 National Strength and Conditioning Association
2476
Copyright © 2020 National Strength and Conditioning Association. Unauthorized reproduction of this article is prohibited.