NE US
Academic Publishers
Advances in Animal and Veterinary Sciences
April 2020 | Volume 8 | Issue 4 | Page 370
INTRODUCTION
C
ancer chemotherapy is considered to be a major
treatment at late stages to avoid the remission of
cancer after surgery (Poornima et al., 2014). It is a typical
methodology of treatment for several types of cancer
(Sahin et al., 2010).
Doxorubicin is one of the most efective anticancer
chemotherapeutic belonging to anthracycline antibiotic
group and it has a large spectrum of activity (Coldwell et
al., 2010). It is being used alone or in combination to treat
a variety of tumors, both hematological and solid, such as
breast cancer ( Jabłonska-Trypuc et al., 2017). Despite its
therapeutic value, doxorubicin has signifcant cardiotoxicity
(Kuznetsova et al., 2011), hepatotoxicity (Patel et al., 2010)
nephrotoxicity (Mohan et al., 2010) and testicular toxicity
(Trivedi et al., 2011) which limit its clinical application.
It also inhibits cell proliferation, induces oxidative stress,
inhibits topoisomerase II, and fnally leads to the cell death
mainly through apoptosis (Ta et al., 2008; Sathesh et al.,
2010; Cao et al., 2013). Although infammation, apoptosis,
mitochondrial DNA damage, impairment of calcium
metabolism and excessive production of free radicals may
all contribute to a variable extent to the deterioration of
organ function, the exact mechanism of doxorubicin-
mediated multiple organ toxicity remains largely unknown
(Gharanei et al., 2014). Doxorubicin tends to accumulate
in mitochondria, causing changes in their structure and
function. However, the main cause of doxorubicin side
Research Article
Abstract | Tis study aims to assess the preventive efects of rutin and/or quercetin on doxorubicin-induced kidney
and heart injuries and oxidative stress in male Wistar rats. Te male Wistar rats, injected with doxorubicin at an
intraperitoneal dose 2 mg/kg b.w. 2 days per week for 5 weeks, were orally treated with rutin and/or quercetin with
dose level 50 mg /kg b.w. every other day for 5weeks. Te treatments of doxorubicin-injected rats with rutin, quercetin
and their combination resulted in a signifcant decrease in the elevated serum creatinine and urea levels refecting
an improvement in kidney function. Similarly, the elevated serum CK-MB and LDH activities were signifcantly
ameliorated as a result of treatments of doxorubicin-injected rats, thereby manifesting an amendment of heart function.
Te treatments also led to the prevention of the elevated lipid peroxidation and amelioration of the lowered GPx,
GST and SOD activities as well as GSH content in kidney and heart as a result of treatment of doxorubicin-injected
rats with rutin and quercetin. Also, the treatments remarkably improved doxorubicin-induced deleterious histological
alterations in kidney and heart. In conclusion, rutin and/or quercetin may have chemopreventive potentials against
doxorubicin-induced nephrocardiotoxicity via suppression of oxidative stress and enhancement of antioxidant defense
system.
Keywords | Rutin, Quercetin, Doxorubicin, Kidney, Heart, Oxidative stress
HEBA UALLAH R. MAHMOUD, OSAMA M. AHMED, HANAA I. FAHIM, NOHA A. AHMED*, MOHAMED
B. ASHOUR
Efects of Rutin and Quercetin on Doxorubicin-Induced
Renocardiotoxicity in Male Wistar Rats
Received | December 05, 2019; Accepted | February 17, 2020; Published | March 20, 2020
*Correspondence | Noha A. Ahmed, Physiology Division, Zoology Department, Faculty of Science, Beni-Suef University, Salah Salim St., 62514, Beni-Suef,
Egypt. Email: drnohascience@science.bsu.edu.eg, drnohascience@gmail.com
Citation | Mahmoud HUR, Ahmed OM, Fahim HI, Ahmed NA, Ashour MB (2020). Efects of rutin and quercetin on doxorubicin-induced renocardiotoxicity
in male wistar rats. Adv. Anim. Vet. Sci. 8(4): 370-384.
DOI | http://dx.doi.org/10.17582/journal.aavs/2020/8.4.370.384
ISSN (Online) | 2307-8316; ISSN (Print) | 2309-3331
Copyright © 2020 Mahmoud et al. Tis is an open access article distributed under the Creative Commons Attribution License, which permits unrestricted use,
distribution, and reproduction in any medium, provided the original work is properly cited.
Physiology Division, Zoology Department, Faculty of Science, Beni-Suef University, P.O. Box 62521, Beni-Suef,
Egypt.