Int. J. Pharm. Sci. Rev. Res., 33(1), July – August 2015; Article No. 13, Pages: 62-67 ISSN 0976 – 044X
International Journal of Pharmaceutical Sciences Review and Research
Available online at www.globalresearchonline.net
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62
Padmaja Kalshetti
a*
, Prasad Thakurdesai
b
, Ramesh Alluri
c
a
Department of Pharmacology, MAEER’S Maharashtra Institute of Pharmacy, Paud Road, Kothrud, Pune, India.
b
Indus Biotech Private Limited, 1, Rahul Residency, Off Salunke Vihar Road, Kondhwa, Pune, India.
c
Dept of Pharmacology, Vishnu Institute of Pharmaceutical Education & Research, Narsapur, Medak District, Andhra Pradesh, India.
* Corresponding author’s E-mail: padmaja.kalshetti@gmail.com
Accepted on: 07-05-2015; Finalized on: 30-06-2015.
ABSTRACT
The main objective of this study was to evaluate the standardized extract of Commiphora mukul Engl. (Burseraceae) in olfactory
bulbectomy induced sexual and immune dysfunction in rats. Olfactory bulbectomy (OBX) was performed in male Sprague dawley
rats (250-270gms). After recovery period of 14 days, 8 groups of animals were made (6 per group) as, Group-I rats served as SHAM
control (Without surgery, burr holes drilled), Group-II rats served as OBX control group, Group-III, IV, V served as standard treatment
groups i.e. imipramine, fluoxetine and desipramine (20mg/ kg p.o., 30mg/ kg p.o., 15mg/ kg p.o.) treated group, Groups VI, VII and VIII
served as drug treatment groups (HECM 50, 100 and 200 mg/ kg p.o.). All the treatments were continued for 14 days after recovery
period. Sexual behaviour parameters were taken on 29
th
day and animals sacrificed at the end for brain dopamine estimation. All
three standards as well as all three doses of hydro alcoholic extract of Commiphora mukul (HECM) does dependently normalized
OBX induced sexual and immune abnormalities. There was a significant improvement in all the parameters of sexual behavior,
altered differential leukocyte count, weight of spleen and thymus and brain DA level by the treatment with standards as well as two
higher doses of HECM. Commiphora mukul at all the doses significantly improved sexual and immune dysfunction induced by OBX,
which is comparable with standard drugs.
Keywords: stress, depression, olfactory bulbectomy, dopamine, sexual dysfunction
INTRODUCTION
epression is a major disorder affecting nearly 13%
- 20% of the world’s population.
1
Roughly, 90% of
depressive patients suffer with mild to moderate
depression, while only 10% are suffering with severely
depression. In case of mild to moderate depression, in
particular, some of the physicians and patients are
reluctant for use of standard antidepressants like
selective serotonin reuptake inhibitors (SSRIs), tricyclic
antidepressants because of their potential and toxic side
effects. Therefore, the additional treatment strategies
with fewer side effects profile, moderate costs and
credible benefits are of particular interest.
2,3
So, in search of new molecules really useful for the
treatment of certain neurological disorders, medicinal
plant research is progressed worldwide by demonstrating
pharmacological effectiveness of various plant species in
a different variety of animal models.
4
Commiphora mukul plant belongs to Burseraceae family
and has a resinous secretion known as guggul. Guggul is
one of the most valuable remedies in ayurvedic system of
medicine. Its usage backs to over 2500 years. Guggul has
been used as antihyperlipidemic, antidiabetic, anti-
inflammatory, antiosteoarthritic, sedative, antispasmodic,
astringent, antiseptic, carminative, expectorant,
emmenagogue, thyroid stimulant, diaphoretic,
antiobesity, diuretic, anthelminitic and demulcent in
traditional medicine. Commiphora mukul has been
reported to contain flavonoids, terpenes, and
phytosterols.
5
However, the steroid guggulsterone has
been purified from the ethylacetate extract of resin.
6
Guggulsterone is the active steroid present in plant and
acts as antagonist of the bile acid farnesoid X receptor, by
demonstrating the hypolipidemic effect of the resin.
The olfactory bulbectomized (OBX) rat is a validated
animal model that meets most of the criteria’s of a
clinical depression. Bilateral removal of the olfactory
bulbs results in a phenotype modeling. Several of the
symptoms seen in major depression, including many of
the behavioral, neurochemical, neuroendocrine and
immune alterations.
7-9
Recently we have reported the antidepressant effects of
standardized extract of commiphora mukul (HECM) in
olfactory bulbectomy induced depression model. It was
found that, HECM represents restorative effects in OBX
induced depression model in rats probably due to stress
reliving mechanisms.
10
Therefore it was found interesting
to study the effect of sub-acute administration of HECM
in olfactory bulbectomy induced sexual dysfunction in
rats.
M ATERIALS AND M ETHODS
Animals
Male Sprague Dawley rats (250–270 g) were purchased
from National Toxicology Centre (NTC), Pune. The animals
were housed at a temperature of 25±1 °C and relative
humidity of 45–55% under 12:12 light: dark cycle. The
animals had free access to feed pellets (Chakan Oil Mills
Effect of Standardized Extract of Commiphora M ukul Engl. ( Burseraceae) on
Bulbectomy Induced Sexual and Immune Dysfunction in Rats.
D
Research Article