Research Article
Protective Effects of Aqueous Extract of Solanum nigrum Linn.
Leaves in Rat Models of Oral Mucositis
Alkesh Patel, Subhankar Biswas, Muhammed Haneefa Shoja,
Grandhi Venkata Ramalingayya, and K. Nandakumar
Department of Pharmacology, Manipal College of Pharmaceutical Sciences, Manipal University, Manipal, Karnataka 576104, India
Correspondence should be addressed to K. Nandakumar; mailnandakumar77@gmail.com
Received 3 July 2014; Revised 30 October 2014; Accepted 30 October 2014; Published 20 November 2014
Academic Editor: Tomas Eferth
Copyright © 2014 Alkesh Patel et al. Tis is an open access article distributed under the Creative Commons Attribution License,
which permits unrestricted use, distribution, and reproduction in any medium, provided the original work is properly cited.
Oral mucositis is one of the most debilitating side efects in patient undergoing chemotherapy or chemoradiotherapy. Leaves of the
plant Solanum nigrum are used in folklore medicine to treat oral ulcers in India. However, no pharmacological investigation has
been carried out till date. Aqueous extract of Solanum nigrum leaves (AESN) was prepared and subjected to various phytochemical
screening. HPLC analysis of the ethyl acetate fraction was carried out. Te aqueous extract (100 and 200 mg/kg) was further
evaluated for its protective efect on two rat models: (a) busulfan plus infrared radiation (chemoradiotherapy) induced oral
mucositis and (b) methotrexate (chemotherapy) induced oral mucositis. Various parameters including body weight change, food
intake, and mortality were measured. AESN showed protective efect in both models of oral mucositis; however, the higher dose
was more efective in chemotherapy induced oral mucositis. A reduction in oral mucositis score ( < 0.05) was observed in the
treatment groups. Signifcant ( < 0.05) improvement in food intake was also observed in AESN treated groups. Aqueous extract
of Solanum nigrum leaves has protective efect on chemotherapy and chemoradiotherapy induced oral mucositis in rats.
1. Introduction
Oral mucositis is a common complication of chemotherapy
and radiotherapy to the head and neck region. It is ofen a
dose limiting toxicity prohibiting the patient from receiving
optimal therapy. Almost every patient with oral cancer
treated with chemoradiotherapy develops deep and painful
wounds characteristic of this condition [1]. Te chance of oral
mucositis occurrence ranges from 30 to 40% in the general
cancer patient population [2]. Conversely, there is a chance
of developing 76% of oral mucositis in patients undergoing
high-dose chemotherapy conditioning before hematopoietic
stem cell transplant [3]. Mucositis is the second most frequent
dose limiting toxicity in patients receiving chemotherapy
[4]. For instance, 40% of patients treated with fuorouracil
based regimens and >60% of patients receiving bone marrow
transplant conditioning therapies for hematological or solid
tumors develop this toxicity [5, 6].
For over a decade, complementary and alternative med-
icine (CAM) has been in use by cancer patients in western
countries (USA, Canada, Germany, etc.) with prevalence
as high as 80% [7, 8]. Among CAM, traditional Chinese
medicine (TCM) is of higher importance, as it is based on
a holistic, natural approach and well established theoretical
framework. Although CAM has potential in treating various
disorders, lack of scientifc data has kept it behind conven-
tional therapies. However, recent studies have investigated
CAM for their potential in alleviating the toxicity associated
with chemotherapy induced mucositis [9]. Here the plant,
Solanum nigrum, commonly known as black nightshade, is
frequently used as a valuable ingredient for clinical TCM
cancer therapy [10]. Chinese people have used the leaves of
this plant to alleviate infammation and edema through its
antipyretic and diuretic efect [11]. Hepatoprotective activity
of this plant is well established [12]. Studies have been
conducted providing evidence for the antitumor potential
of this plant, including liver, stomach, lung, bladder, breast,
and colon cancer [10]. Leaves of this plant have been used as
traditional folk medicine by the inhabitants of southern India
to treat mouth ulcers. To our knowledge, no study has been
conducted to determine the protective efect of this plant for
oral mucositis. Terefore, the purpose of this study was aimed
Hindawi Publishing Corporation
e Scientific World Journal
Volume 2014, Article ID 345939, 10 pages
http://dx.doi.org/10.1155/2014/345939