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The Pharma Innovation Journal 2023; 12(2): 2442-2448
ISSN (E): 2277-7695
ISSN (P): 2349-8242
NAAS Rating: 5.23
TPI 2023; 12(2): 2442-2448
© 2023 TPI
www.thepharmajournal.com
Received: 21-11-2022
Accepted: 24-12-2022
Pulagurtha Bhaskararao
(1) Associate Professor, Aditya
Pharmacy College, Surampalem,
Andhra Pradesh, India
(2)
)
Jawaharlal Nehru
Technological University
Kakinada, Kakinada, Andhra
Pradesh, India
Kontham Venkataramanapa
Raju
(1) Aditya Pharmacy College,
Surampalem, Andhra Pradesh,
India
(2)
)
Jawaharlal Nehru
Technological University
Kakinada, Kakinada, Andhra
Pradesh, India
Balla Sujiya
(1) Aditya Pharmacy College,
Surampalem, Andhra Pradesh,
India
(2)
)
Jawaharlal Nehru
Technological University
Kakinada, Kakinada, Andhra
Pradesh, India
Corresponding Author:
Pulagurtha Bhaskararao
(1) Associate Professor, Aditya
Pharmacy College, Surampalem,
Andhra Pradesh, India
(2)
)
Jawaharlal Nehru
Technological University
Kakinada, Kakinada, Andhra
Pradesh, India
Method development and validation for the
simultaneous estimation of amlodipine besylate and
atorvastatin calcium in pharmaceutical dosage forms
by micellar liquid chromatography
Pulagurtha Bhaskararao, Kontham Venkataramanapa Raju and Balla
Sujiya
Abstract
The present study is aimed at developing and validating an accurate, precise, linear and robust micellar
liquid chromatographic method for the simultaneous estimation of amlodipine besylate (AB) and
atorvastatin calcium (AC) in pharmaceutical dosage forms. The analysis of AB and AC is done with a
mixture of n-butanol and polysorbate 20 (0.05 M) in the ratio of 30:70 (v/v) as mobile phase and
Phenomenex C18 column (150 mm × 4.6 mm, 5 μm) as stationary phase. The chromatographic peaks of
AB and AC were detected and measured at 240 nm. The retention times of AB and AC were found to be
3.61 min and 6.53 min, respectively. The developed method is demonstrated to access its suitability for
meeting its intended purpose by the validation with a set of validation parameters as per ICH and USP
guidelines. The method is proved to be linear from 5 to 50 μg/ml for AB and 10 to 100 μg/ml for AC
with the correlation coefficients of 0.9995 and 0.9990, respectively. The method is found to be precise
with percent relative standard deviation value in range 0.8-1.1% and 0.5-1.0% and accurate with
recoveries of 99.20 to 101.20% and 98.80 to 100.67% for AB and AC respectively.
Keywords: Amlodipine besylate, atorvastatin calcium, polysorbate 20, micellar liquid chromatography,
stability indicating, analysis
Introduction
Amlodipine besylate (AB), chemically called as (3-ethyl 5-methyl 2-[(2aminoethoxy o
methyl]-4-(2chlorophenyl)-methyl 1,4 dihydropyridine,3,5dihydrocarboxylate), is a
dihydropyridine and long-acting potent calcium channel blocker used for the treatment of
hypertension, congestive heart failure and angina pectoris
[1]
. AB lowers the blood pressure,
relaxes the heart muscles and dilates the heart blood vessels to prevent spasm
[2, 3]
. Chemical
structure of AB is given in Fig 1. Atorvastatin calcium (AC), described chemically as ([R-(R*,
R*)]-2-(4-fluorophenyl)-β, δ-dihydroxy-5-(1-methylethyl)-3-phenyl-4-[(phenylamino)
carbonyl] -1H-pyrrole-1-heptanoic acid, calcium salt (2:1) trihydrate). AC is an
antihyperlipidemic agent belonging to drug class statins
[3]
. AC is widely used in the treatment
of hypercholesterolemia. AC decreases the levels of low-density lipoproteins and triglycerides
to a major extent and slightly increases the level of high-density lipoprotein
[4]
. Chemical
structure of AC is given in Fig 1.
Fig 1: Structure of amlodipine besylate and atorvastatin calcium