Toxicology Letters 96,97 (1998) 245 – 251 Defense and repair mechanisms in the airway epithelium exposed to oxidative stress Effects of analogues of retinoic acid Armelle Baeza-Squiban *, Emmanuelle Boisvieux-Ulrich, Laure Delcher, Francelyne Marano Laboratoire de Cytophysiologie et Toxicologie cellulaire, Uniersite ´ Paris 7, Denis Diderot, tour 53 -54, 3 e ´tage, case 7073, 2 place jussieu, 75 251 Paris ce ´dex 05, France Abstract A model of rabbit tracheal epithelial (RTE) cells in vitro was developed in order to investigate the effects, on the airway epithelium, of reactive oxygen species (ROS) generated by H 2 O 2 in association or not in association with Fe 2 + . The immediate consequence of a 24 h exposure of RTE cells to an oxidative stress was an increase in catalase activity whereas superoxide dismutase activity was not modified. A latter consequence of a chronic ROS insult was the induction of a repair mechanism which led to squamous metaplasia (SM). SM is characterized by a stratification of the epithelium, the expression of the cytokeratin 13 and the appearance of cells with cross-linked envelopes. Reversible modifications between mucociliary and squamous phenotype are modulated by retinoids. The action of retinoids is selective: metaplasia is inhibited by agonists of RARand receptors and not by an agonist of RAR receptors. © 1998 Elsevier Science Ireland Ltd. All rights reserved. Keywords: Tracheal epithelium; Oxidative stress; Squamous metaplasia; Anti-oxidant enzymes; Retinoids 1. Introduction The respiratory tract is continually exposed to air pollutants which are frequently present in urban atmosphere. Epidemiological studies have demonstrated that environmental pollution is im- plicated in the maintenance and/or aggravation of pre-existing respiratory diseases. Many atmo- spheric pollutants are oxidants as O 3 , NO 2 , SO 2 , some mineral particles and components of cigarette smoke (Weitzman and Graceffa, 1984; Schlesinger, 1989; Mossman et al., 1990; Guil- ianelli et al., 1993; Chitano et al., 1995). In addi- tion to their oxidative properties, these pollutants may secondarily activate macrophages and neu- trophiles to release reactive oxygen species (ROS) (Barnes, 1990). In vivo studies have not clarified * Corresponding author. Tel.: +33 01 44276062; fax: +33 01 44276999; e-mail: Marano@paris7.jussieu.fr 0378-4274/98/$19.00 © 1998 Elsevier Science Ireland Ltd. All rights reserved. PII S0378-4274(98)00079-4